SCHEMBL765844

SCHEMBL765844

NOc1ccc(Oc2ccc(CNC(=O)C3(NC(=O)c4ccnnc4)CC3)cc2)c(C(F)(F)F)c1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BDKRB1 P46663 2/20 0.42
CNR1 P21554 1/20 0.36
MAPK14 Q16539 3/20 0.35
PTGER4 P35408 2/20 0.35
PTGER2 P43116 1/20 0.35
DDR2 Q16832 2/20 0.33
SUCNR1 Q9BXA5 1/20 0.33
MAPK11 Q15759 1/20 0.32
CYP3A4 P08684 1/20 0.32
SCD O00767 1/20 0.32
CCR2 P41597 1/20 0.32
F10 P00742 1/20 0.32
MAPT P10636 1/20 0.32
TP53 P04637 1/20 0.32
MDM2 Q00987 1/20 0.32
HTR2C P28335 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL765643 0.92 BDKRB1 (0.45) BDKRB1CNR1F10MAPT
SCHEMBL765818 0.89 BDKRB1 (0.41) BDKRB1MAPK14PTGER4PTGER2DDR2
SCHEMBL10121214 0.87 BDKRB1 (0.40) BDKRB1MAPK14PTGER4PTGER2DDR2
SCHEMBL10121216 0.84 BDKRB1 (0.41) BDKRB1MAPK14PTGER4PTGER2SUCNR1
SCHEMBL10121111 0.83 BDKRB1 (0.37) BDKRB1MAPK14PTGER4PTGER2CYP3A4
SCHEMBL13191643 0.83 P2RX7 (0.39) BDKRB1F10MAPT
SCHEMBL12238926 0.82 BDKRB1 (0.49) BDKRB1
SCHEMBL10121524 0.82 BDKRB1 (0.44) BDKRB1F10
SCHEMBL765551 0.81 BDKRB1 (0.35) BDKRB1MAPK14PTGER4PTGER2CYP3A4
SCHEMBL764476 0.81 BDKRB1 (0.35) BDKRB1MAPK14PTGER4PTGER2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2188254-B1 NOVEL BRADYKININ B1-ANTAGONISTS BOEHRINGER INGELHEIM INT (DE) 2012-03-21 EP disclosed