SCHEMBL7658901

SCHEMBL7658901

C[C@@H]1OC(=O)N(C(=O)NCCCN2CCC(c3ccc(F)cc3)CC2)[C@H]1c1ccc(F)c(F)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 18/20 1.00
ADRA1B P35368 17/20 1.00
ADRA1D P25100 16/20 1.00
HRH1 P35367 3/20 1.00
ADRA2A P08913 2/20 0.58
ADRA2B P18089 2/20 0.58
ADRA2C P18825 2/20 0.58
CCR2 P41597 1/20 0.46
CCR3 P51677 1/20 0.46
MCHR1 Q99705 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6954383 1.00 ADRA1A (1.00) ADRA1AADRA1BADRA1DHRH1ADRA2A
SCHEMBL14587407 0.94 ADRA1A (0.89) ADRA1AADRA1BADRA1DHRH1ADRA2A
SCHEMBL6961810 0.90 ADRA1A (0.82) ADRA1AADRA1BADRA1DHRH1ADRA2A
SCHEMBL7226018 0.89 ADRA1A (0.80) ADRA1AADRA1BADRA1DHRH1ADRA2A
SCHEMBL5663201 0.87 ADRA1A (0.76) ADRA1AADRA1BADRA1DHRH1MCHR1
SCHEMBL7068045 0.87 ADRA1A (0.76) ADRA1AADRA1BADRA1DHRH1MCHR1
SCHEMBL7068048 0.87 ADRA1A (0.76) ADRA1AADRA1BADRA1DHRH1MCHR1
SCHEMBL7966480 0.84 ADRA1A (0.72) ADRA1AADRA1BADRA1DHRH1ADRA2A
SCHEMBL7952342 0.84 ADRA1A (0.72) ADRA1AADRA1BADRA1DHRH1ADRA2A
SCHEMBL7952365 0.84 ADRA1A (0.72) ADRA1AADRA1BADRA1DHRH1ADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6372911-B1 REACTING COMPOUND CONTAINING AT LEAST ONE CARBON-CARBON DOUBLE BOND WITH CARBAMATE IN AQUEOUS SOLVENT IN PRESENCE OF BASE, OSMIUM CATALYST, CO-OXIDANT, AND OPTIONALLY ASYMMETRIC LIGAND, TO FORM REACTION MIXTURE CONTAINING BETA-HYDROXY CARBAMATE MERCK & CO., INC. 2002-04-16 US disclosed
US-6329393-B1 ADRENERGIC AGENTS TREATMENT OF BENIGN PROSTATIC HYPERPLASIA. MERCK & CO., INC. 2001-12-11 US disclosed