SCHEMBL7656532

SCHEMBL7656532

CC(C)c1ccc(C(=O)Nc2ccc3c(c2)CN(C)C(C)(C)C3)cc1C#N

nearest known ligand 0.43

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 10/20 0.43
NAMPT P43490 5/20 0.40
L3MBTL3 Q96JM7 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7656595 0.86 ROCK2 (0.39) ROCK2NAMPT
SCHEMBL6295077 0.84 ROCK2 (0.58) ROCK2
Hydrochloric Acid SCHEMBL6299497 0.83 ROCK2 (0.57) ROCK2
SCHEMBL7993332 0.83 ROCK2 (0.45) ROCK2NAMPT
SCHEMBL7653872 0.82 ROCK2 (0.38) ROCK2
SCHEMBL7659472 0.81 ROCK2 (0.43) ROCK2
SCHEMBL7659848 0.77 ROCK2 (0.39) ROCK2NAMPTL3MBTL3
SCHEMBL7656812 0.76 CYP26A1 (0.38) ROCK2
SCHEMBL7655629 0.76 ROCK2 (0.50) ROCK2
SCHEMBL6806888 0.75 ROCK2 (0.38) ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6492378-B1 Substituted isoquinoline derivatives and their use as anticonvulsivants SMITHKLINE BEECHAM P.L.C. (GB) 2002-12-10 US claimed
US-6492378-B1 Substituted isoquinoline derivatives and their use as anticonvulsivants SMITHKLINE BEECHAM P.L.C. (GB) 2002-12-10 US disclosed