SCHEMBL7659537

SCHEMBL7659537

CCOC(=O)N1CCN(C(=O)NC(CS(=O)(=O)Cc2ccccc2)C(=O)NCC#N)CC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 2/20 0.51
GAA P10253 1/20 0.51
TSHR P16473 1/20 0.51
CTSS P25774 10/20 0.47
CTSB P07858 5/20 0.47
CTSL P07711 5/20 0.47
MAPT P10636 2/20 0.46
CTSK P43235 4/20 0.44
L3MBTL1 Q9Y468 1/20 0.43
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
POLB P06746 1/20 0.42
GFER P55789 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
MEN1 O00255 1/20 0.42
USP2 O75604 1/20 0.42
ALDH1A1 P00352 1/20 0.42
CASP1 P29466 1/20 0.42
HBB P68871 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6742147 0.89 CTSS (0.51) CTSSCTSBCTSLCTSK
SCHEMBL6744248 0.83 ALDH1A1 (0.54) TSHRCTSSCTSBCTSLCYP2D6
SCHEMBL5523222 0.82 NPC1 (0.53) CYP2C19CTSSCTSBCTSLMAPT
SCHEMBL7659544 0.82 GAA (0.54) CYP2C19GAATSHRMAPTL3MBTL1
SCHEMBL6742702 0.81 CTSS (0.43) CTSSCTSBCTSLCTSKL3MBTL1
SCHEMBL6742158 0.78 CTSS (0.68) CTSSCTSBCTSLCTSK
SCHEMBL6061195 0.78 CTSS (0.68) CTSSCTSBCTSLCTSK
SCHEMBL6740685 0.77 CTSS (0.55) GAACTSSCTSBCTSLL3MBTL1
SCHEMBL6740689 0.77 CTSS (0.55) GAACTSSCTSBCTSLL3MBTL1
SCHEMBL6738423 0.76 CTSS (0.77) CTSSCTSBCTSLCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6492362-B1 Compounds and compositions as cathepsin S inhibitors AXYS PHARMACEUTICALS, INC. 2002-12-10 US disclosed