SCHEMBL7659544

SCHEMBL7659544

CCOC(=O)N1CCN(C(=O)NCC(C(=O)NCC#N)S(=O)(=O)Cc2ccccc2)CC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.54
TSHR P16473 2/20 0.54
CYP2C19 P33261 1/20 0.54
MAPT P10636 3/20 0.48
SMN1; SMN2 Q16637 3/20 0.46
RORC P51449 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.45
ALDH1A1 P00352 3/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
USP2 O75604 1/20 0.44
CASP1 P29466 1/20 0.44
HBB P68871 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
POLB P06746 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C9 P11712 1/20 0.43
ABL1 P00519 1/20 0.43
RIN1 Q13671 1/20 0.43
TDP1 Q9NUW8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6742152 0.88 STS (0.50)
SCHEMBL6744961 0.85 CTSS (0.48)
SCHEMBL6744250 0.82 ALDH1A1 (0.52) GAACYP2C19ALDH1A1USP2NPSR1
SCHEMBL5523231 0.82 ALDH1A1 (0.56) GAATSHRCYP2C19MAPTSMN1; SMN2
SCHEMBL7659537 0.82 CYP2C19 (0.51) GAATSHRCYP2C19MAPTSMN1; SMN2
SCHEMBL6742707 0.77 TSHR (0.50) GAATSHRCYP2C19MAPTSMN1; SMN2
SCHEMBL6740690 0.77 CTSS (0.45) GAAL3MBTL1
SCHEMBL6061910 0.75 CTSL (0.56)
SCHEMBL5523222 0.74 NPC1 (0.53) CYP2C19MAPTSMN1; SMN2L3MBTL1ALDH1A1
SCHEMBL6741766 0.73 CTSS (0.60)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6492362-B1 Compounds and compositions as cathepsin S inhibitors AXYS PHARMACEUTICALS, INC. 2002-12-10 US disclosed