SCHEMBL7659667

SCHEMBL7659667

CCOC(=O)c1nc(-c2cccnc2)no1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.60
NPC1 O15118 7/20 0.55
SMN1; SMN2 Q16637 6/20 0.55
RAB9A P51151 6/20 0.55
MAPT P10636 6/20 0.55
TP53 P04637 4/20 0.55
LMNA P02545 1/20 0.55
KMT2A Q03164 1/20 0.55
NFKB1 P19838 2/20 0.54
NFKB2 Q00653 2/20 0.54
RELA Q04206 2/20 0.54
S1PR1 P21453 2/20 0.52
PKM P14618 1/20 0.52
DCTPP1 Q9H773 1/20 0.52
CHRNB2 P17787 1/20 0.51
CHRNA5 P30532 1/20 0.51
CHRNA4 P43681 1/20 0.51
NPSR1 Q6W5P4 2/20 0.51
ALDH1A1 P00352 1/20 0.51
PPARA Q07869 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2554648 0.85 HTT (0.67) HTTNPC1SMN1; SMN2RAB9AMAPT
SCHEMBL4528391 0.84 HTT (0.66) HTTNPC1SMN1; SMN2RAB9AMAPT
SCHEMBL27768478 0.81 CHRNB2 (0.63) NPC1SMN1; SMN2RAB9AMAPTTP53
SCHEMBL3233714 0.80 HTT (0.71) HTTNPC1SMN1; SMN2RAB9AMAPT
SCHEMBL3419014 0.80 NPC1 (0.52) HTTNPC1SMN1; SMN2RAB9AMAPT
SCHEMBL4751192 0.80 HTT (0.67) HTTSMN1; SMN2MAPTLMNAKMT2A
SCHEMBL1815822 0.79 CHRNB2 (0.61) NPC1SMN1; SMN2RAB9AMAPTTP53
SCHEMBL17476086 0.79 HTT (0.59) HTTNPC1SMN1; SMN2RAB9AMAPT
SCHEMBL22619755 0.79 HTT (0.66) HTTNPC1SMN1; SMN2RAB9AMAPT
SCHEMBL31039805 0.79 HTT (0.66) HTTNPC1SMN1; SMN2RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6465462-B1 COGNITION ENHANCEMENT FOR DEMENTING ILLNESSES SUCH AS ALZHEIMER'S DISEASE MERCK SHARP & DOHME LTD. 2002-10-15 US disclosed