SCHEMBL27768478

SCHEMBL27768478

O=C(c1nc(-c2cccnc2)no1)c1nc(-c2cccnc2)no1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.63
CHRNA5 P30532 2/20 0.63
CHRNA4 P43681 2/20 0.63
SMN1; SMN2 Q16637 6/20 0.56
NPC1 O15118 6/20 0.56
RAB9A P51151 6/20 0.56
TP53 P04637 5/20 0.56
ALDH1A1 P00352 5/20 0.56
MAPT P10636 3/20 0.56
KDM4E B2RXH2 2/20 0.56
HPGD P15428 2/20 0.56
HSD17B10 Q99714 1/20 0.56
PPARA Q07869 6/20 0.55
PKM P14618 1/20 0.54
TSHR P16473 3/20 0.54
NPSR1 Q6W5P4 2/20 0.54
POLB P06746 1/20 0.54
NFKB1 P19838 1/20 0.54
NFKB2 Q00653 1/20 0.54
RELA Q04206 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1815822 0.89 CHRNB2 (0.61) CHRNB2CHRNA5CHRNA4SMN1; SMN2NPC1
SCHEMBL3418996 0.84 GAA (0.57) CHRNB2CHRNA5CHRNA4SMN1; SMN2NPC1
SCHEMBL1432036 0.84 MKNK1 (0.57) CHRNB2CHRNA5CHRNA4SMN1; SMN2NPC1
SCHEMBL27768533 0.81 NR1H4 (0.57) SMN1; SMN2NPC1RAB9ATP53ALDH1A1
SCHEMBL3419014 0.81 NPC1 (0.52) CHRNB2CHRNA5CHRNA4SMN1; SMN2NPC1
SCHEMBL7659667 0.81 HTT (0.60) CHRNB2CHRNA5CHRNA4SMN1; SMN2NPC1
SCHEMBL27789974 0.80 MAPT (0.56) SMN1; SMN2NPC1RAB9ATP53ALDH1A1
SCHEMBL1422890 0.78 CHRNB2 (1.00) CHRNB2CHRNA5CHRNA4SMN1; SMN2NPC1
SCHEMBL4313968 0.76 RAB9A (0.59) CHRNB2CHRNA5CHRNA4SMN1; SMN2NPC1
SCHEMBL14427066 0.75 NPC1 (0.47) CHRNB2CHRNA5CHRNA4SMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102850324-A Indole compounds MICROBIA INC 2013-01-02 CN disclosed
CN-101563337-A Indole compounds MICROBIA INC (US) 2009-10-21 CN disclosed