SCHEMBL7659713

SCHEMBL7659713

COc1cc(OC(C)C)c(Cl)cc1C(=O)Nc1cccc2c1C(C)(C)CNC2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.42
POLB P06746 2/20 0.42
CASP3 P42574 1/20 0.42
ATM Q13315 1/20 0.42
SENP8 Q96LD8 1/20 0.42
SENP7 Q9BQF6 1/20 0.42
SENP6 Q9GZR1 1/20 0.42
KDM4E B2RXH2 4/20 0.41
ALDH1A1 P00352 4/20 0.41
KMT2A Q03164 3/20 0.41
MAPT P10636 4/20 0.38
LMNA P02545 4/20 0.38
HTT P42858 2/20 0.38
BRPF1 P55201 1/20 0.38
PTGS2 P35354 1/20 0.38
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
TOP1 P11387 2/20 0.37
RXFP1 Q9HBX9 1/20 0.37
RAB9A P51151 4/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7658672 0.84 KMT2A (0.42) NPC1POLBCASP3ATMSENP8
SCHEMBL8186096 0.74 ROCK2 (0.46) NPC1POLBCASP3ATMSENP8
SCHEMBL8185203 0.74 KMT2A (0.48) NPC1POLBCASP3ATMSENP8
SCHEMBL7991365 0.70 BRPF1 (0.43) NPC1POLBCASP3ATMSENP8
SCHEMBL8176080 0.68 KMT2A (0.51) NPC1POLBCASP3ATMSENP8
Hydrochloric Acid SCHEMBL8186121 0.67 KMT2A (0.50) NPC1POLBCASP3ATMSENP8
SCHEMBL8174320 0.67 NPC1 (0.43) NPC1POLBCASP3ATMSENP8
SCHEMBL6806468 0.67 ROCK2 (0.36) NPC1KMT2AMAPTBRPF1RXFP1
SCHEMBL8176053 0.66 ROCK2 (0.59) NPC1KMT2AMAPTRAB9ASMN1; SMN2
Hydrochloric Acid SCHEMBL6810196 0.66 ROCK2 (0.36) NPC1KMT2AMAPTBRPF1RXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6492378-B1 Substituted isoquinoline derivatives and their use as anticonvulsivants SMITHKLINE BEECHAM P.L.C. (GB) 2002-12-10 US disclosed
EP-1104404-A1 SUBSTITUTED ISOQUINOLINE DERIVATIVES AND THEIR USE AS ANTICONVULSANTS SMITHKLINE BEECHAM PLC (GB) 2001-06-06 EP disclosed
WO-2000009486-A1 SUBSTITUTED ISOQUINOLINE DERIVATIVES AND THEIR USE AS ANTICONVULSIVANTS SMITHKLINE BEECHAM P.L.C. (GB) 2000-02-24 WO disclosed