SCHEMBL7662930

SCHEMBL7662930

O=C(O)C(=O)CC(=O)c1cccc(Cn2cnc3ccccc32)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 3/20 0.58
CYP11B2 P19099 3/20 0.58
TNF P01375 1/20 0.57
IDO1 P14902 9/20 0.55
ALDH1A1 P00352 1/20 0.55
HDAC1 Q13547 1/20 0.54
HDAC6 Q9UBN7 1/20 0.54
HRH3 Q9Y5N1 1/20 0.52
CA12 O43570 1/20 0.52
CA1 P00915 1/20 0.52
CA2 P00918 1/20 0.52
CA7 P43166 1/20 0.52
CA9 Q16790 1/20 0.52
CA13 Q8N1Q1 1/20 0.52
CDYL2 Q8N8U2 1/20 0.50
CDYL Q9Y232 1/20 0.50
CDY1; CDY1B Q9Y6F8 1/20 0.50
PTPN1 P18031 1/20 0.50
LMNA P02545 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2885662 0.85 CYP11B1 (0.67) CYP11B1CYP11B2TNFIDO1ALDH1A1
SCHEMBL7668846 0.81 CYP11B1 (0.53) CYP11B1CYP11B2TNFIDO1ALDH1A1
SCHEMBL13085846 0.81 IDO1 (0.64) CYP11B1CYP11B2TNFIDO1ALDH1A1
SCHEMBL6950593 0.79 FEN1 (0.57) HDAC1HDAC6PTPN1SMN1; SMN2
SCHEMBL7667737 0.79 GRM2 (0.57) ALDH1A1PTPN1LMNASMN1; SMN2
SCHEMBL31722842 0.78 CYP11B1 (0.80) CYP11B1CYP11B2TNFIDO1ALDH1A1
SCHEMBL3177643 0.78 CYP11B1 (0.80) CYP11B1CYP11B2TNFIDO1ALDH1A1
SCHEMBL9303119 0.77 FAAH (0.60) CYP11B1CYP11B2IDO1ALDH1A1HDAC1
SCHEMBL9302980 0.77 CYP11B1 (0.62) CYP11B1CYP11B2TNFIDO1ALDH1A1
SCHEMBL230002 0.75 CYP11B1 (1.00) CYP11B1CYP11B2TNFALDH1A1HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US claimed
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US disclosed