SCHEMBL7662978

SCHEMBL7662978

COc1ccc(C(=O)O)cc1S(=O)(=O)NCCN1CCOCC1

nearest known ligand 0.72

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.72
MAPT P10636 2/20 0.64
PKM P14618 2/20 0.61
POLB P06746 1/20 0.61
ALDH1A1 P00352 2/20 0.61
KDM4E B2RXH2 1/20 0.54
KMT2A Q03164 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
CYP2D6 P10635 1/20 0.53
CYP2C9 P11712 1/20 0.53
TSHR P16473 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15765534 0.94 SMN1; SMN2 (0.63) SMN1; SMN2MAPTPKMPOLBALDH1A1
SCHEMBL15754508 0.92 SMN1; SMN2 (0.72) SMN1; SMN2MAPTPKMALDH1A1KMT2A
SCHEMBL20240486 0.82 SMN1; SMN2 (0.73) SMN1; SMN2MAPTPKMALDH1A1KMT2A
SCHEMBL7676271 0.82 SMN1; SMN2 (0.58) SMN1; SMN2MAPTALDH1A1KDM4EKMT2A
SCHEMBL4616589 0.81 SMN1; SMN2 (0.69) SMN1; SMN2PKMPOLBALDH1A1KMT2A
SCHEMBL8073771 0.81 KMT2A (0.58) SMN1; SMN2PKMPOLBALDH1A1KMT2A
SCHEMBL18830935 0.80 CYP2C9 (0.56) SMN1; SMN2MAPTPOLBALDH1A1KDM4E
SCHEMBL20240439 0.80 SMN1; SMN2 (0.75) SMN1; SMN2PKMALDH1A1KMT2ATSHR
SCHEMBL8019642 0.80 SMN1; SMN2 (0.56) SMN1; SMN2MAPTALDH1A1KDM4EKMT2A
SCHEMBL7663344 0.80 SMN1; SMN2 (0.56) SMN1; SMN2MAPTALDH1A1KDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110698459-B 1-phenyl-2-pyridylalkyl alcohol derivatives as phosphodiesterase inhibitors 奇斯药制品公司 2023-05-05 CN disclosed
CN-110698459-A 1-phenyl-2-pyridylalkyl alcohol derivatives as phosphodiesterase inhibitors 奇斯药制品公司 2020-01-17 CN disclosed
US-9944612-B2 1-phenyl-2-pyridinyl alkyl alcohol derivatives as phosphodiesterase inhibitors CHIESI FARMACEUTICI S.P.A. (IT) 2018-04-17 US disclosed
US-9944612-B2 1-phenyl-2-pyridinyl alkyl alcohol derivatives as phosphodiesterase inhibitors CHIESI FARMACEUTICI S.P.A. (IT) 2018-04-17 US disclosed
US-9944612-B2 1-phenyl-2-pyridinyl alkyl alcohol derivatives as phosphodiesterase inhibitors CHIESI FARMACEUTICI S.P.A. (IT) 2018-04-17 US disclosed
EP-2928869-A1 1-PHENYL-2-PYRIDINYL ALKYL ALCOHOL DERIVATIVES AS PHOSPHODIESTERASE INHIBITORS Chiesi Farmaceutici S.p.A. (IT) 2015-10-14 EP disclosed
WO-2014086865-A1 1-PHENYL-2-PYRIDINYL ALKYL ALCOHOL DERIVATIVES AS PHOSPHODIESTERASE INHIBITORS CHIESI FARMACEUTICI S.P.A. (IT) 2014-06-12 WO disclosed
WO-2014086865-A1 1-PHENYL-2-PYRIDINYL ALKYL ALCOHOL DERIVATIVES AS PHOSPHODIESTERASE INHIBITORS CHIESI FARMACEUTICI S.P.A. (IT) 2014-06-12 WO disclosed
US-20140155391-A1 1-PHENYL-2-PYRIDINYL ALKYL ALCOHOL DERIVATIVES AS PHOSPHODIESTERASE INHIBITORS CHIESI FARMACEUTICI S.P.A. (IT) 2014-06-05 US disclosed
US-20140155391-A1 1-PHENYL-2-PYRIDINYL ALKYL ALCOHOL DERIVATIVES AS PHOSPHODIESTERASE INHIBITORS CHIESI FARMACEUTICI S.P.A. (IT) 2014-06-05 US disclosed
US-20140155391-A1 1-PHENYL-2-PYRIDINYL ALKYL ALCOHOL DERIVATIVES AS PHOSPHODIESTERASE INHIBITORS CHIESI FARMACEUTICI S.P.A. (IT) 2014-06-05 US disclosed
US-20020111369-A1 Aryl sulfonic acids and derivatives as FSH antagonists AMERICAN HOME PRODUCTS CORPORATION (US) 2002-08-15 US disclosed
US-6355633-B1 CONTRACEPTIVES AMERICAN HOME PRODUCTS CORPORATION 2002-03-12 US disclosed
WO-2000058277-A1 ARYL SULFONIC ACIDS AND DERIVATIVES AS FSH ANTAGONISTS AMERICAN HOME PRODUCTS CORPORATION (US) 2000-10-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140155391-A1 1-PHENYL-2-PYRIDINYL ALKYL ALCOHOL DERIVATIVES AS PHOSPHODIESTERASE INHIBITORS PDE4A, PDE4B, PDE3A SMN1; SMN2 2901/4885MAPT 4037/4885PKM 1567/4885
US-20020111369-A1 Aryl sulfonic acids and derivatives as FSH antagonists FSHR, GNRHR, LHCGR SMN1; SMN2 2927/4885MAPT 4858/4885PKM 4553/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.