SCHEMBL7663

SCHEMBL7663

COc1ccc(NCC2CCN(C(=O)C3CC3)C2)c([N+](=O)[O-])c1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.51
RECQL P46063 2/20 0.51
LMNA P02545 1/20 0.50
MAPT P10636 6/20 0.48
HPGD P15428 1/20 0.48
TRPV1 Q8NER1 1/20 0.48
MAPK1 P28482 3/20 0.48
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
AKR1C3 P42330 2/20 0.45
AKR1C2 P52895 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7661 1.00 ALDH1A1 (0.51) ALDH1A1RECQLLMNAMAPTHPGD
SCHEMBL5748 0.92 ALDH1A1 (0.48) ALDH1A1RECQLLMNAMAPTHPGD
SCHEMBL5746 0.92 ALDH1A1 (0.48) ALDH1A1RECQLLMNAMAPTHPGD
SCHEMBL11909636 0.90 ALDH1A1 (0.52) ALDH1A1RECQLLMNAMAPTHPGD
SCHEMBL11909631 0.90 ALDH1A1 (0.52) ALDH1A1RECQLLMNAMAPTHPGD
SCHEMBL6263 0.87 KAT2B (0.44) ALDH1A1LMNAMAPTTRPV1MEN1
SCHEMBL6261 0.87 KAT2B (0.44) ALDH1A1LMNAMAPTTRPV1MEN1
SCHEMBL5904 0.85 NPY5R (0.42) MAPTMAPK1KMT2A
SCHEMBL5906 0.85 NPY5R (0.42) MAPTMAPK1KMT2A
SCHEMBL10321 0.84 ALDH1A1 (0.48) ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2493310-A1 BENZIMIDAZOLES AS FATTY ACID SYNTHASE INHIBITORS GlaxoSmithKline LLC (US) 2012-09-05 EP disclosed
WO-2011056635-A1 BENZIMIDAZOLES AS FATTY ACID SYNTHASE INHIBITORS GLAXOSMITHKLINE LLC (US) 2011-05-12 WO disclosed