SCHEMBL7664922

SCHEMBL7664922

CC(C)c1c[nH]c(Cc2ccccc2)n1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 2/20 0.43
GAA P10253 1/20 0.41
NR1H2 P55055 1/20 0.40
NR1H3 Q13133 1/20 0.40
NPC1 O15118 1/20 0.40
POLB P06746 1/20 0.40
RAB9A P51151 1/20 0.40
HRH3 Q9Y5N1 1/20 0.40
ADORA2A P29274 2/20 0.38
ADORA1 P30542 2/20 0.38
KMT2A Q03164 1/20 0.38
CAPN1 P07384 1/20 0.38
CALM1 P0DP23 1/20 0.37
DAO P14920 1/20 0.37
LMNA P02545 1/20 0.36
HSD17B10 Q99714 1/20 0.36
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4903117 0.81 TSHR (0.46) HRH3KMT2ALMNATSHR
SCHEMBL316101 0.78 TAAR1 (0.48) TAAR1GAANR1H2NR1H3NPC1
SCHEMBL1723556 0.78 TAAR1 (0.48) TAAR1GAANR1H2NR1H3NPC1
SCHEMBL6971912 0.75 HRH3 (0.51) HRH3KMT2ATSHR
SCHEMBL24787891 0.74 RIPK1 (0.40) TAAR1
SCHEMBL3695497 0.74 DDAH1 (0.31) ADORA2AADORA1
SCHEMBL5850108 0.73 KDM4E (0.42) GAANPC1POLBRAB9AKMT2A
SCHEMBL10650713 0.73 TAAR1 (0.47) TAAR1GAANR1H2NR1H3NPC1
SCHEMBL7936430 0.73 TAAR1 (0.47) TAAR1GAANR1H2NR1H3NPC1
SCHEMBL5469222 0.73 TAAR1 (0.47) TAAR1GAANR1H2NR1H3NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6492377-B1 Imidazotriazolopyrimidines with adenosine-antagonistic activity BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-12-10 US disclosed