SCHEMBL6971912

SCHEMBL6971912

CC(C)c1c[nH]c(CCCOCc2ccccc2)n1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 4/20 0.51
HRH4 Q9H3N8 3/20 0.51
L3MBTL1 Q9Y468 2/20 0.40
TDP1 Q9NUW8 1/20 0.40
ALDH1A1 P00352 2/20 0.36
TSHR P16473 1/20 0.36
SOAT1 P35610 1/20 0.34
HTT P42858 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.33
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4901240 0.92 HRH4 (0.44) HRH3HRH4L3MBTL1TDP1ALDH1A1
SCHEMBL4903117 0.85 TSHR (0.46) HRH3HRH4ALDH1A1TSHRHTT
SCHEMBL7664922 0.75 TAAR1 (0.43) HRH3TSHRKMT2A
SCHEMBL6962088 0.74 HRH4 (0.43) HRH3HRH4L3MBTL1TDP1ALDH1A1
SCHEMBL4893200 0.71 HRH4 (0.45) HRH3HRH4L3MBTL1TDP1ALDH1A1
SCHEMBL6966941 0.70 IDO1 (0.42) L3MBTL1TDP1ALDH1A1HTTSMN1; SMN2
SCHEMBL4069939 0.69 TDP1 (0.64) HRH3HRH4L3MBTL1TDP1TSHR
Proxyfan SCHEMBL15929504 0.68 HRH3 (1.00) HRH3HRH4
SCHEMBL7479206 0.68 HRH3 (0.44) HRH3HRH4L3MBTL1TDP1ALDH1A1
SCHEMBL7474823 0.68 HRH4 (0.44) HRH3HRH4L3MBTL1TDP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed