SCHEMBL7665154

SCHEMBL7665154

CC(Cc1ccnc2ccccc12)(C(=O)NC(CO)Cc1ccccc1)N(C(=O)O)C1C2CC3CC(C2)CC1C3

nearest known ligand 0.41

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 1/20 0.35
PARP1 P09874 1/20 0.35
PARP3 Q9Y6F1 1/20 0.35
CCR1 P32246 1/20 0.35
CYP3A4 P08684 1/20 0.35
MAPK1 P28482 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7666814 0.88 NPY1R (0.37) CCKBRCYP3A4MAPK1
SCHEMBL6897076 0.84 CCKBR (0.51) CCKBR
SCHEMBL6897079 0.84 CCKBR (0.51) CCKBR
SCHEMBL7664606 0.81 CYP3A4 (0.38) CYP3A4MAPK1
SCHEMBL7667464 0.79 CYP3A4 (0.34) CCKBRCYP3A4MAPK1
SCHEMBL7664675 0.78 NPY5R (0.32) CCKBR
SCHEMBL9698405 0.76 KDM4E (0.45) PARP1PARP3CCR1CYP3A4MAPK1
SCHEMBL9699591 0.72 CCKBR (0.43) CCKBR
SCHEMBL7667387 0.70 CCKBR (0.46) CCKBR
SCHEMBL7662981 0.69 EPHX2 (0.39) CCKBRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993003721-A1 CHOLECYSTOKININ ANTAGONISTS USEFUL FOR TREATING DEPRESSION WARNER-LAMBERT COMPANY (US) 1993-03-04 WO claimed
US-6492531-B1 THE INVENTION CONCERNS CHOLECYSTOKININ (CCK) ANTAGONISTS USEFUL IN THE TREATMENT OF COGNITIVE DISORDERS. ESPECIALLY USEFUL ARE CCK.SUB.B ANTAGONISTS SUCH AS CI-988. WARNER-LAMBERT COMPANY 2002-12-10 US disclosed