SCHEMBL7664606

SCHEMBL7664606

CC(Cc1ccc2ccccc2c1)(C(=O)NC(CO)Cc1ccccc1)N(C(=O)O)C1C2CC3CC(C2)CC1C3

nearest known ligand 0.39

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.38
MAPK1 P28482 1/20 0.38
MME P08473 2/20 0.36
CASR P41180 1/20 0.36
PIN1 Q13526 1/20 0.35
ACE P12821 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7666814 0.86 NPY1R (0.37) CYP3A4MAPK1
SCHEMBL7667767 0.82 EPHX2 (0.44)
SCHEMBL6897076 0.81 CCKBR (0.51)
SCHEMBL7665154 0.81 CCKBR (0.35) CYP3A4MAPK1
SCHEMBL6897079 0.81 CCKBR (0.51)
SCHEMBL7667464 0.80 CYP3A4 (0.34) CYP3A4MAPK1
SCHEMBL7670952 0.78 ALDH1A1 (0.38)
SCHEMBL7664675 0.77 NPY5R (0.32)
SCHEMBL7662981 0.72 EPHX2 (0.39) MAPK1
SCHEMBL9698370 0.71 CCKBR (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993003721-A1 CHOLECYSTOKININ ANTAGONISTS USEFUL FOR TREATING DEPRESSION WARNER-LAMBERT COMPANY (US) 1993-03-04 WO claimed
US-6492531-B1 THE INVENTION CONCERNS CHOLECYSTOKININ (CCK) ANTAGONISTS USEFUL IN THE TREATMENT OF COGNITIVE DISORDERS. ESPECIALLY USEFUL ARE CCK.SUB.B ANTAGONISTS SUCH AS CI-988. WARNER-LAMBERT COMPANY 2002-12-10 US disclosed