SCHEMBL7666173

SCHEMBL7666173

CC(C)(C)[C@](CCC(N)=O)(NC(=O)c1ccc(NC(Cn2ccnc2)c2ccc(F)cc2)cc1-c1ccccc1)C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.44
CYP51A1 Q16850 6/20 0.41
AURKA O14965 1/20 0.40
PDPK1 O15530 1/20 0.40
RPS6KB1 P23443 1/20 0.40
CYP3A4 P08684 5/20 0.39
CYP2C19 P33261 4/20 0.39
CYP2D6 P10635 2/20 0.39
CYP2C9 P11712 2/20 0.39
FNTA P49354 1/20 0.38
FNTB P49356 1/20 0.38
PGGT1B P53609 1/20 0.38
CYP1A2 P05177 1/20 0.36
CYP26A1 O43174 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7660603 0.87 PTGS2 (0.40) PTGS2CYP51A1AURKAPDPK1RPS6KB1
SCHEMBL7659533 0.83 CYP51A1 (0.46) PTGS2CYP51A1AURKAPDPK1RPS6KB1
SCHEMBL7667482 0.83 PTGS2 (0.43) PTGS2CYP51A1CYP3A4CYP2C19CYP2D6
SCHEMBL7666164 0.82 CYP3A4 (0.45) PTGS2CYP51A1CYP3A4CYP2C19CYP2D6
SCHEMBL7666171 0.80 FNTA (0.49) PTGS2CYP51A1AURKAPDPK1RPS6KB1
SCHEMBL7656241 0.79 CYP51A1 (0.40) PTGS2CYP51A1CYP3A4CYP2C19CYP2D6
SCHEMBL7662081 0.79 CYP51A1 (0.40) PTGS2CYP51A1AURKAPDPK1RPS6KB1
SCHEMBL7669388 0.77 CYP51A1 (0.40) PTGS2CYP51A1CYP3A4CYP2C19CYP2D6
SCHEMBL7656582 0.77 CYP51A1 (0.49) PTGS2CYP51A1AURKAPDPK1RPS6KB1
SCHEMBL7660388 0.76 FNTA (0.56) FNTAFNTBPGGT1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6410539-B1 ANTICARCINOGENIC AGENTS ASTRAZENCA UK LIMITED (GB) 2002-06-25 US claimed