SCHEMBL7666649

SCHEMBL7666649

COc1n[nH]c(=O)n1Cc1cc(-c2ccccc2)ccc1C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 4/20 0.39
P2RX7 Q99572 2/20 0.39
KDM4E B2RXH2 2/20 0.38
GAA P10253 2/20 0.38
MAPT P10636 2/20 0.38
HPGD P15428 2/20 0.38
PRMT5 O14744 1/20 0.36
CYP1A2 P05177 1/20 0.35
FAAH O00519 1/20 0.35
MGLL Q99685 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HTT P42858 1/20 0.35
AGTR1 P30556 1/20 0.35
AGTR2 P50052 1/20 0.35
TNKS2 Q9H2K2 1/20 0.35
BACE1 P56817 1/20 0.35
PDE4A P27815 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4C Q08493 1/20 0.34
PDE4D Q08499 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7671424 0.89 CCNC (0.42) CHEK1MAPTALDH1A1
SCHEMBL7667237 0.86 KDM4E (0.40) CHEK1KDM4EHPGDPRMT5TNKS2
SCHEMBL6776723 0.82 AGTR1 (0.43) CHEK1KDM4EHPGDPRMT5CYP1A2
SCHEMBL7671615 0.81 HPGD (0.41) P2RX7KDM4EGAAMAPTHPGD
SCHEMBL7666760 0.80 ALDH1A1 (0.43) CHEK1KDM4EMAPTPRMT5ALDH1A1
SCHEMBL7668981 0.74 CHEK1 (0.38) CHEK1P2RX7KDM4EHPGDCYP1A2
SCHEMBL7666815 0.72 HPGD (0.44) MAPTHPGDCYP1A2HTT
SCHEMBL7669141 0.72 TP53 (0.44) KDM4EGAAMAPTHPGDALDH1A1
SCHEMBL7672496 0.71 TP53 (0.41) KDM4EGAAMAPTHPGDALDH1A1
SCHEMBL7671400 0.71 TP53 (0.41) CHEK1MAPTHPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6489487-B1 AGRICULTURAL OR HORTICULTURAL FUNGICIDES SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2002-12-03 US disclosed
EP-1103548-A1 TRIAZOLONE DERIVATIVES, USE THEREOF, AND INTERMEDIATE THEREFOR SUMITOMO CHEMICAL COMPANY LIMITED (JP) 2001-05-30 EP disclosed