SCHEMBL7667196

SCHEMBL7667196

CC(=O)NCc1cc(OC[C@@H]2CCN2C(=O)OC(C)(C)C)cnc1Cl

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.42
ALOX5AP P20292 3/20 0.36
FEN1 P39748 1/20 0.36
GPR119 Q8TDV5 4/20 0.35
EPHX2 P34913 1/20 0.35
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
CHRNA7 P36544 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6585968 0.96 ALDH1A1 (0.39) ALDH1A1ALOX5APFEN1GPR119EPHX2
SCHEMBL7676310 0.93 ALDH1A1 (0.42) ALDH1A1ALOX5APFEN1GPR119EPHX2
SCHEMBL6584996 0.91 ALDH1A1 (0.41) ALDH1A1ALOX5APFEN1GPR119EPHX2
SCHEMBL7478777 0.88 ALOX5AP (0.39) ALDH1A1ALOX5APFEN1GPR119CHRNB4
SCHEMBL6587429 0.88 KDM4E (0.45) ALDH1A1ALOX5AP
SCHEMBL7134497 0.87 CHRNA3 (0.39) ALDH1A1ALOX5APFEN1GPR119CHRNB4
SCHEMBL6584732 0.86 ALOX5AP (0.39) ALDH1A1ALOX5APFEN1GPR119CHRNB4
SCHEMBL6585517 0.85 MAPT (0.40) ALDH1A1
SCHEMBL7470605 0.84 ALOX5AP (0.41) ALDH1A1ALOX5APFEN1GPR119CHRNB4
SCHEMBL7667587 0.84 ALOX5AP (0.37) ALDH1A1ALOX5APFEN1GPR119CHRNB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6437138-B1 5-BROMO-6-CHLORO-3-(2-(S)-AZETIDINYL OR PYRROLIDINYL-METHOXY) PYRIDINE INTERMEDIATES FOR THE 5-SUBSTITUTED COMPOUNDS WHICH ARE POTENT LIGANDS AT NEURONAL NICOTINIC CHOLINERGIC CHANNEL RECEPTORS, NEUROTRANSMITTER CONTROLLING AGENTS ABBOTT LABORATORIES 2002-08-20 US disclosed
US-6127386-A STIMULANTS, NEUROTRANSMITTERS, CHOLINERGIC AGENTS ABBOTT LABORATORIES (US) 2000-10-03 US disclosed