SCHEMBL6587429

SCHEMBL6587429

CC(C)(C)OC(=O)N1CC[C@H]1COc1cnc(Cl)c(CNC(=O)c2ccccc2)c1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.45
PKM P14618 1/20 0.45
HDAC1 Q13547 2/20 0.41
ALDH1A1 P00352 1/20 0.40
MAPK8 P45983 2/20 0.40
NR1H2 P55055 1/20 0.39
LMNA P02545 1/20 0.38
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
ALOX5AP P20292 2/20 0.37
TP53 P04637 1/20 0.37
ACACB O00763 1/20 0.37
ACACA Q13085 1/20 0.37
USP30 Q70CQ3 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6585455 0.93 KDM4E (0.40) KDM4EPKMHDAC1ALDH1A1MAPK8
SCHEMBL6585151 0.88 L3MBTL1 (0.42) KDM4EALDH1A1LMNA
SCHEMBL7676310 0.88 ALDH1A1 (0.42) ALDH1A1ALOX5AP
SCHEMBL7667196 0.88 ALDH1A1 (0.42) ALDH1A1ALOX5AP
SCHEMBL6585517 0.87 MAPT (0.40) HDAC1ALDH1A1TP53
SCHEMBL6584996 0.86 ALDH1A1 (0.41) ALDH1A1ALOX5AP
SCHEMBL6582165 0.86 CHRNA3 (0.49)
SCHEMBL6583669 0.85 KDM4E (0.40) KDM4EPKMALOX5AP
Hydrochloric Acid SCHEMBL6588512 0.85 CHRNA3 (0.48)
SCHEMBL6585968 0.84 ALDH1A1 (0.39) ALDH1A1ALOX5AP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0934308-B1 3-PYRIDYLOXYMETHYL HETEROCYCLIC ETHER COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION ABBOTT LAB (US) 2004-08-11 EP disclosed
US-6437138-B1 5-BROMO-6-CHLORO-3-(2-(S)-AZETIDINYL OR PYRROLIDINYL-METHOXY) PYRIDINE INTERMEDIATES FOR THE 5-SUBSTITUTED COMPOUNDS WHICH ARE POTENT LIGANDS AT NEURONAL NICOTINIC CHOLINERGIC CHANNEL RECEPTORS, NEUROTRANSMITTER CONTROLLING AGENTS ABBOTT LABORATORIES 2002-08-20 US disclosed
US-6127386-A STIMULANTS, NEUROTRANSMITTERS, CHOLINERGIC AGENTS ABBOTT LABORATORIES (US) 2000-10-03 US disclosed
US-5629325-A TREATMENT OF NERVOUS SYSTEM DISORDERS; NEURONAL NICOTINIC CHOLINERGIC COMPOUNDS ABBOTT LABORATORIES (US) 1997-05-13 US disclosed