SCHEMBL7667724

SCHEMBL7667724

CCn1c(=O)c2c(nc(C(C)(C)C)n2CCN2CCOCC2)n2nc(Cc3ccc(O)cc3)nc12

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RXFP1 Q9HBX9 1/20 0.35
ALDH1A1 P00352 5/20 0.35
HTT P42858 4/20 0.35
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
BRD4 O60885 1/20 0.35
CREBBP Q92793 1/20 0.35
GAA P10253 2/20 0.35
MAPK1 P28482 2/20 0.34
HSD17B10 Q99714 1/20 0.34
PDE5A O76074 2/20 0.33
USP2 O75604 1/20 0.33
LMNA P02545 1/20 0.33
TSHR P16473 1/20 0.33
CNR2 P34972 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7667529 0.84 ADORA2A (0.38) ADORA2AADORA1PDE5A
SCHEMBL7002349 0.71 ADORA2B (0.38) ADORA2AADORA1
SCHEMBL7760161 0.63 ADORA3 (0.50) ALDH1A1HTTADORA2AADORA1MAPK1
SCHEMBL23235098 0.58 SIGMAR1 (0.60) HTTCYP2C9HSD17B10
SCHEMBL8348067 0.55 GAA (0.55) ALDH1A1GAAMAPK1HSD17B10TSHR
SCHEMBL4024799 0.55 HRH3 (0.71) ALDH1A1HTTCYP2C9HSD17B10LMNA
SCHEMBL5321100 0.54 ATM (0.58) ALDH1A1HTTMAPK1TSHR
SCHEMBL25217971 0.54 RXFP1 (0.63) RXFP1ALDH1A1CYP3A4CYP2C9GAA
SCHEMBL27550438 0.53 CYP2D6 (0.57) ALDH1A1HTTCYP3A4CYP2C9LMNA
SCHEMBL8563151 0.53 SIGMAR1 (0.42) ALDH1A1CYP3A4CYP2C9MAPK1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6492377-B1 Imidazotriazolopyrimidines with adenosine-antagonistic activity BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-12-10 US disclosed