SCHEMBL7668693

SCHEMBL7668693

CCn1c(=O)c2[nH]c(C3CCCC3)nc2n2nc(Cc3ccc(F)c(F)c3)nc12

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 8/20 0.51
ADORA2A P29274 4/20 0.51
ADORA2B P29275 4/20 0.51
ADORA3 P0DMS8 3/20 0.51
MEN1 O00255 1/20 0.45
GMNN O75496 1/20 0.45
LMNA P02545 1/20 0.45
CYP1A2 P05177 1/20 0.45
TSHR P16473 1/20 0.45
PMP22 Q01453 1/20 0.45
KMT2A Q03164 1/20 0.45
HIF1A Q16665 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7668320 0.90 ADORA1 (0.53) ADORA1ADORA2AADORA2BADORA3MEN1
SCHEMBL7662113 0.82 ADORA1 (0.51) ADORA1ADORA2AADORA2BADORA3MEN1
SCHEMBL7003429 0.81 ADORA1 (0.58) ADORA1ADORA2AADORA2BADORA3MEN1
SCHEMBL6998057 0.81 ADORA1 (0.58) ADORA1ADORA2AADORA2BADORA3MEN1
SCHEMBL7002301 0.81 ADORA1 (0.61) ADORA1ADORA2AADORA2BADORA3MEN1
SCHEMBL7656557 0.81 ADORA3 (0.58) ADORA1ADORA2AADORA2BADORA3MEN1
SCHEMBL7666406 0.80 ADORA3 (0.51) ADORA1ADORA2AADORA2BADORA3MEN1
SCHEMBL7661349 0.79 ADORA2A (0.58) ADORA1ADORA2AADORA2BADORA3MEN1
SCHEMBL6997855 0.79 ADORA1 (0.55) ADORA1ADORA2AADORA2BADORA3MEN1
SCHEMBL7662109 0.78 ADORA1 (0.48) ADORA1ADORA2AADORA2BADORA3MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6492377-B1 Imidazotriazolopyrimidines with adenosine-antagonistic activity BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-12-10 US disclosed