SCHEMBL7669074

SCHEMBL7669074

COc1ccc(-c2ccnc3ccccc23)cc1OC

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACACA Q13085 1/20 0.59
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
ACVR1 Q04771 3/20 0.51
AAK1 Q2M2I8 3/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
ERN1 O75460 1/20 0.49
KDM4E B2RXH2 2/20 0.49
NPC1 O15118 2/20 0.49
ALDH1A1 P00352 2/20 0.49
HPGD P15428 1/20 0.49
GUSB P08236 1/20 0.49
RAB9A P51151 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
ABCG2 Q9UNQ0 3/20 0.48
ABCB1 P08183 1/20 0.47
ABCC1 P33527 1/20 0.47
GAK O14976 1/20 0.47
RIPK2 O43353 1/20 0.47
COQ8A Q8NI60 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23496991 0.88 TLR8 (0.53) ACACAACVR1AAK1ERN1GAK
SCHEMBL12989150 0.87 CYP1A1 (0.52) ACACAMEN1KMT2AACVR1AAK1
SCHEMBL7418556 0.85 PDE4A (0.54)
SCHEMBL11822911 0.84 PDGFRB (0.57) ACVR1GAKRIPK2COQ8ANLK
SCHEMBL11808233 0.81 TLR8 (0.60) ACACAAAK1NPC1SMN1; SMN2GAK
SCHEMBL16549179 0.81 KIT (0.48) MEN1KMT2AL3MBTL1KDM4EALDH1A1
SCHEMBL30251801 0.80 BMP4 (0.61) ACACAMEN1KMT2AACVR1L3MBTL1
SCHEMBL7665284 0.80 BMP4 (0.61) ACACAMEN1KMT2AACVR1L3MBTL1
SCHEMBL27290306 0.79 CLK4 (0.53) ACACAKMT2AACVR1ALDH1A1HPGD
SCHEMBL29269603 0.78 ALDH1A1 (0.51) ACVR1KDM4ENPC1ALDH1A1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6388081-B1 4-substituted-quinoline derivatives and 4-substituted-quinoline combinatorial libraries LION BIOSCIENCE AG (DE) 2002-05-14 US disclosed
US-6262269-B1 4-Substituted-quinoline derivatives and 4-substituted-quinoline combinatorial libraries TREGA BIOSCIENCES, INC. 2001-07-17 US disclosed
EP-0977989-A1 4-SUBSTITUTED-QUINOLINE DERIVATIVES AND 4-SUBSTITUTE-QUINOLINE COMBINATORIAL LIBRARIES TREGA BIOSCIENCES, INC. (US) 2000-02-09 EP disclosed
WO-1998034115-A1 4-SUBSTITUTED-QUINOLINE DERIVATIVES AND 4-SUBSTITUTE-QUINOLINE COMBINATORIAL LIBRARIES TREGA BIOSCIENCES, INC. (US) 1998-08-06 WO disclosed
US-3936461-A Substituted 4-benzylquinolines WARNER-LAMBERT COMPANY (US) 1976-02-03 US disclosed