SCHEMBL7669302

SCHEMBL7669302

CCc1nc2c([nH]1)c(=O)n(CC)c1nc(CC3CCCCC3)nn21

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 5/20 0.53
ADORA2B P29275 5/20 0.53
ADORA1 P30542 6/20 0.51
ADORA3 P0DMS8 2/20 0.41
PDE9A O76083 2/20 0.36
PDE1C Q14123 1/20 0.36
MEN1 O00255 1/20 0.35
GMNN O75496 1/20 0.35
LMNA P02545 1/20 0.35
CYP1A2 P05177 1/20 0.35
TSHR P16473 1/20 0.35
PMP22 Q01453 1/20 0.35
KMT2A Q03164 1/20 0.35
HIF1A Q16665 1/20 0.35
CDK1 P06493 1/20 0.34
CCNB1 P14635 1/20 0.34
CCNA2 P20248 1/20 0.34
CDK2 P24941 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8563310 0.92 ADORA2A (0.53) ADORA2AADORA2BADORA1ADORA3PDE9A
SCHEMBL7661349 0.86 ADORA2A (0.58) ADORA2AADORA2BADORA1ADORA3MEN1
SCHEMBL7669942 0.82 ADORA2A (0.47) ADORA2AADORA2BADORA1ADORA3
SCHEMBL7669969 0.79 ADORA1 (0.40) ADORA2AADORA2BADORA1ADORA3MEN1
SCHEMBL7671399 0.79 ADORA1 (0.40) ADORA2AADORA2BADORA1ADORA3MEN1
SCHEMBL8560943 0.77 ADORA2A (0.46) ADORA2AADORA2BADORA1
SCHEMBL7671625 0.74 ADORA2B (0.46) ADORA2AADORA2BADORA1ADORA3CYP1A2
SCHEMBL7002301 0.73 ADORA1 (0.61) ADORA2AADORA2BADORA1ADORA3MEN1
SCHEMBL7671642 0.72 ADORA2A (0.42) ADORA2AADORA2BADORA1ADORA3CDK1
SCHEMBL7665749 0.72 ADORA2B (0.43) ADORA2AADORA2BADORA1ADORA3CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6492377-B1 Imidazotriazolopyrimidines with adenosine-antagonistic activity BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-12-10 US disclosed