SCHEMBL8563310

SCHEMBL8563310

CCc1nc2c([nH]1)c(=O)n1nc(CC3CCCCC3)nc1n2CC

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 5/20 0.53
ADORA2B P29275 5/20 0.53
ADORA1 P30542 6/20 0.51
ADORA3 P0DMS8 2/20 0.41
PDE9A O76083 2/20 0.36
PDE1C Q14123 1/20 0.36
MEN1 O00255 1/20 0.35
GMNN O75496 1/20 0.35
LMNA P02545 1/20 0.35
CYP1A2 P05177 1/20 0.35
TSHR P16473 1/20 0.35
PMP22 Q01453 1/20 0.35
KMT2A Q03164 1/20 0.35
HIF1A Q16665 1/20 0.35
CDK1 P06493 1/20 0.34
CCNB1 P14635 1/20 0.34
CCNA2 P20248 1/20 0.34
CDK2 P24941 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7669302 0.92 ADORA2A (0.53) ADORA2AADORA2BADORA1ADORA3PDE9A
SCHEMBL8560943 0.81 ADORA2A (0.46) ADORA2AADORA2BADORA1
SCHEMBL7661349 0.78 ADORA2A (0.58) ADORA2AADORA2BADORA1ADORA3MEN1
SCHEMBL7669942 0.75 ADORA2A (0.47) ADORA2AADORA2BADORA1ADORA3
SCHEMBL8558501 0.75 ADORA1 (0.45) ADORA2AADORA2BADORA1
SCHEMBL8559224 0.73 ADORA1 (0.61) ADORA2AADORA2BADORA1ADORA3MEN1
SCHEMBL7671399 0.71 ADORA1 (0.40) ADORA2AADORA2BADORA1ADORA3MEN1
SCHEMBL7669969 0.71 ADORA1 (0.40) ADORA2AADORA2BADORA1ADORA3MEN1
SCHEMBL8562980 0.71 ADORA1 (0.57) ADORA2AADORA2BADORA1ADORA3MEN1
SCHEMBL11021594 0.68 ADORA2A (0.53) ADORA2AADORA2BADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0880524-A1 NEW TRIAZOLOPURINES, METHOD OF PREPARING THEM AND THEIR USE AS DRUGS Boehringer Ingelheim Pharma KG (DE) 1998-12-02 EP disclosed
WO-1998003511-A1 NEW TRIAZOLOPURINES, METHOD OF PREPARING THEM AND THEIR USE AS DRUGS BOEHRINGER INGELHEIM PHARMA KG (DE) 1998-01-29 WO disclosed