SCHEMBL8560943

SCHEMBL8560943

CCn1c2nc[nH]c2c(=O)n2nc(CC3CCCCC3)nc12

nearest known ligand 0.46

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 14/20 0.46
ADORA2B P29275 11/20 0.46
PDE4A P27815 12/20 0.44
PDE4B Q07343 12/20 0.44
PDE4C Q08493 12/20 0.44
PDE4D Q08499 12/20 0.44
ADORA1 P30542 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7669942 0.93 ADORA2A (0.47) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL8563310 0.81 ADORA2A (0.53) ADORA2AADORA2BADORA1
SCHEMBL7669302 0.77 ADORA2A (0.53) ADORA2AADORA2BADORA1
SCHEMBL7661349 0.76 ADORA2A (0.58) ADORA2AADORA2BADORA1
SCHEMBL7669969 0.71 ADORA1 (0.40) ADORA2AADORA2BADORA1
SCHEMBL7671399 0.71 ADORA1 (0.40) ADORA2AADORA2BADORA1
SCHEMBL8560750 0.69 PDE4A (0.52) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL7025705 0.68 ADORA2B (0.55) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL5005966 0.68 ADORA2A (0.62) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL7666660 0.67 ADORA2B (0.54) ADORA2AADORA2BPDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0880524-A1 NEW TRIAZOLOPURINES, METHOD OF PREPARING THEM AND THEIR USE AS DRUGS Boehringer Ingelheim Pharma KG (DE) 1998-12-02 EP disclosed
WO-1998003511-A1 NEW TRIAZOLOPURINES, METHOD OF PREPARING THEM AND THEIR USE AS DRUGS BOEHRINGER INGELHEIM PHARMA KG (DE) 1998-01-29 WO disclosed