SCHEMBL7671402

SCHEMBL7671402

CCn1c(=O)c2[nH]c(C34CC5CC(CC3C5)C4)nc2n2nc(Cc3cccnc3)nc12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 5/20 0.50
ADORA2A P29274 5/20 0.50
ADORA2B P29275 5/20 0.50
ADORA3 P0DMS8 5/20 0.50
SLC6A3 Q01959 1/20 0.50
SLC22A6 Q4U2R8 1/20 0.50
SLC22A8 Q8TCC7 1/20 0.50
SLC22A11 Q9NSA0 1/20 0.50
MEN1 O00255 1/20 0.46
MAPT P10636 1/20 0.46
KMT2A Q03164 1/20 0.46
HSD11B1 P28845 2/20 0.33
CYP17A1 P05093 3/20 0.33
CYP19A1 P11511 3/20 0.33
CCNB2 O95067 1/20 0.32
CCNE2 O96020 1/20 0.32
CDK1 P06493 1/20 0.32
CDK4 P11802 1/20 0.32
CCNB1 P14635 1/20 0.32
CCND1 P24385 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7664157 0.91 ADORA2B (0.54) ADORA1ADORA2AADORA2BADORA3SLC6A3
SCHEMBL7671642 0.79 ADORA2A (0.42) ADORA1ADORA2AADORA2BADORA3CCNB2
SCHEMBL7662113 0.78 ADORA1 (0.51) ADORA1ADORA2AADORA2BADORA3MEN1
SCHEMBL7665201 0.75 ADORA2A (0.45) ADORA2AADORA2BADORA3KMT2A
SCHEMBL7668670 0.73 ADORA2B (0.51) ADORA1ADORA2AADORA2BADORA3MEN1
SCHEMBL7269103 0.72 ADORA1 (0.81) ADORA1ADORA2AADORA2BADORA3SLC6A3
SCHEMBL8203454 0.71 ADORA1 (0.80) ADORA1ADORA2AADORA2BADORA3SLC6A3
SCHEMBL14051422 0.70 ADORA1 (0.91) ADORA1ADORA2AADORA2BADORA3SLC6A3
SCHEMBL8203432 0.70 ADORA1 (0.78) ADORA1ADORA2AADORA2BADORA3SLC6A3
SCHEMBL7670431 0.68 ADORA2B (0.54) ADORA1ADORA2AADORA2BADORA3MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6492377-B1 Imidazotriazolopyrimidines with adenosine-antagonistic activity BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-12-10 US disclosed