SCHEMBL7664157

SCHEMBL7664157

CCn1c(=O)c2[nH]c(C34CC5CC(CC3C5)C4)nc2n2nc(Cc3ccccc3)nc12

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 8/20 0.54
ADORA2A P29274 7/20 0.54
ADORA1 P30542 6/20 0.54
ADORA3 P0DMS8 6/20 0.54
SLC6A3 Q01959 1/20 0.54
SLC22A6 Q4U2R8 1/20 0.54
SLC22A8 Q8TCC7 1/20 0.54
SLC22A11 Q9NSA0 1/20 0.54
MEN1 O00255 1/20 0.49
MAPT P10636 1/20 0.49
KMT2A Q03164 1/20 0.49
SIRT1 Q96EB6 1/20 0.35
SIRT3 Q9NTG7 1/20 0.35
SIRT5 Q9NXA8 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
HPGD P15428 1/20 0.35
TSHR P16473 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7671402 0.91 ADORA1 (0.50) ADORA2BADORA2AADORA1ADORA3SLC6A3
SCHEMBL8203454 0.78 ADORA1 (0.80) ADORA2BADORA2AADORA1ADORA3SLC6A3
SCHEMBL8203432 0.76 ADORA1 (0.78) ADORA2BADORA2AADORA1ADORA3SLC6A3
SCHEMBL7269103 0.76 ADORA1 (0.81) ADORA2BADORA2AADORA1ADORA3SLC6A3
SCHEMBL7666682 0.74 ADORA3 (0.50) ADORA2BADORA2AADORA1ADORA3MEN1
SCHEMBL14051422 0.73 ADORA1 (0.91) ADORA2BADORA2AADORA1ADORA3SLC6A3
SCHEMBL7670431 0.73 ADORA2B (0.54) ADORA2BADORA2AADORA1ADORA3MEN1
SCHEMBL7666680 0.73 ADORA3 (0.47) ADORA2BADORA2AADORA1ADORA3MEN1
SCHEMBL7659412 0.72 ADORA2B (0.45) ADORA2BADORA2AADORA1ADORA3MEN1
SCHEMBL6999142 0.72 SIRT1 (0.46) ADORA2BADORA2AADORA1ADORA3MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6492377-B1 Imidazotriazolopyrimidines with adenosine-antagonistic activity BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-12-10 US disclosed