SCHEMBL7674124

SCHEMBL7674124

O=C(Cl)c1cccnc1Oc1cccc(Cl)c1

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.58
POLB P06746 1/20 0.58
GAA P10253 1/20 0.58
RAB9A P51151 1/20 0.55
TDP1 Q9NUW8 1/20 0.49
P2RY1 P47900 1/20 0.47
PTGER4 P35408 1/20 0.46
PDE4A P27815 1/20 0.46
PDE4B Q07343 1/20 0.46
PDE4C Q08493 1/20 0.46
PDE4D Q08499 1/20 0.46
MAPK8 P45983 2/20 0.45
ADRB3 P13945 1/20 0.44
CYP1A2 P05177 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
KDM4E B2RXH2 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2332693 0.89 ALDH1A1 (0.61) ALDH1A1POLBGAARAB9ATDP1
SCHEMBL7364681 0.87 RAB9A (0.72) ALDH1A1POLBGAARAB9ATDP1
SCHEMBL29209327 0.84 TDP1 (0.51) ALDH1A1POLBGAARAB9ATDP1
SCHEMBL30749506 0.84 TDP1 (0.51) ALDH1A1POLBGAARAB9ATDP1
SCHEMBL2924686 0.84 RAB9A (0.76) ALDH1A1POLBGAARAB9ATDP1
SCHEMBL1086604 0.83 ALDH1A1 (0.70) ALDH1A1POLBGAARAB9ATDP1
SCHEMBL27565178 0.83 RAB9A (0.55) ALDH1A1POLBGAARAB9ATDP1
SCHEMBL3454297 0.82 CYP1A2 (0.62) ALDH1A1POLBGAARAB9ATDP1
SCHEMBL8177633 0.81 KDM4E (0.62) P2RY1CYP1A2CYP2C9CYP2C19KDM4E
SCHEMBL11247603 0.81 NPC1 (0.63) ALDH1A1POLBGAARAB9AP2RY1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6380218-B1 FOR THERAPY OF RESPIRATORY, ALLERGIC, AND INFLAMMATORY DISORDERS COMPRISING ASTHMA, CHRONIC OBSTRUCTIVE PULMONARY DISEASE, ACUTE RESPIRATORY DISEASE SYNDROME, PULMONARY HYPERSENSITIVITY, AND ALLERGIC RHINITIS IN A MAMMAL PFIZER INC 2002-04-30 US disclosed
CN-1254335-A Nicotinamide derivatives PFIZER PROD INC (US) 2000-05-24 CN disclosed
US-4327218-A HERBICIDES STAUFFER CHEMICAL COMPANY (US) 1982-04-27 US disclosed
US-4270946-A N-Aryl,2-phenoxy nicotinamide compounds and the herbicidal use thereof STAUFFER CHEMICAL COMPANY (US) 1981-06-02 US disclosed
US-4251263-A N-substituted, 2-phenoxynicotinamide compounds and the herbicidal use thereof STAUFFER CHEMICAL COMPANY (US) 1981-02-17 US disclosed