SCHEMBL7678633

SCHEMBL7678633

CCC1=CCC(C)(C)c2cc(C)c(Nc3ccc(C(=O)O)c(CC)c3)cc21

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA P19793 5/20 0.35
TAS2R14 Q9NYV8 1/20 0.34
RARB P10826 3/20 0.33
RARA P10276 2/20 0.33
RARG P13631 2/20 0.33
PTGS1 P23219 1/20 0.33
PTGS2 P35354 1/20 0.33
RXRB P28702 1/20 0.32
RXRG P48443 1/20 0.32
CYP26A1 O43174 1/20 0.32
CYP26B1 Q9NR63 1/20 0.32
AKR1C3 P42330 4/20 0.32
AKR1C2 P52895 4/20 0.32
CLCN2 P51788 1/20 0.32
MEN1 O00255 2/20 0.31
MAPT P10636 2/20 0.31
KMT2A Q03164 2/20 0.31
GAA P10253 1/20 0.31
AKR1B10 O60218 1/20 0.31
AKR1B1 P15121 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6087117 0.76 MEN1 (0.43) MEN1MAPTKMT2AGAA
SCHEMBL6086582 0.73 RARB (0.46) RXRARARBRARARARGRXRB
SCHEMBL7695986 0.72 MEN1 (0.42) MEN1MAPTKMT2AGAA
SCHEMBL8771863 0.70 RARB (0.51) RXRARARBRARARARG
SCHEMBL22836931 0.67 RARB (0.60) RXRARARBRARARARGRXRB
SCHEMBL7699420 0.67 CLCN2 (0.43) TAS2R14RARBRARARARGPTGS1
SCHEMBL4654712 0.67 RARA (0.59) RXRARARBRARARARGCYP26A1
SCHEMBL6086727 0.66 RAB9A (0.42) MEN1MAPTKMT2AGAALMNA
SCHEMBL6715212 0.66 RXRA (0.66) RXRARARBRARARARGRXRB
SCHEMBL9141154 0.65 MAPT (0.51) AKR1C3AKR1C2CLCN2MEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1265848-A2 AMINES SUBSTITUTED WITH A DIHYDRONAPHTHALENYL, CRHOMENYL, OR THIOCHROMENYL GROUP, AN ARYL OR HETEROARYL GROUP AND AN ALKYL GROUP, HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY Allergan Sales, Inc. (US) 2002-12-18 EP disclosed
WO-2001070668-A2 AMINES SUBSTITUTED WITH A DIHYDRONAPHTHALENYL, CRHOMENYL, OR THIOCHROMENYL GROUP, AN ARYL OR HETEROARYL GROUP AND AN ALKYL GROUP, HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY ALLERGAN, INC. (US) 2001-09-27 WO disclosed