SCHEMBL7680686

SCHEMBL7680686

CN1CCCN(C2CCCc3cc(C=O)ccc32)CC1

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.46
MEN1 O00255 1/20 0.46
GAA P10253 1/20 0.46
MAPT P10636 1/20 0.46
HPGD P15428 1/20 0.46
KMT2A Q03164 1/20 0.46
CHRNA7 P36544 1/20 0.40
MTNR1B P49286 2/20 0.38
ALDH1A3 P47895 3/20 0.37
HTR2C P28335 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28064840 0.88 ALDH1A1 (0.44) ALDH1A1MEN1GAAMAPTHPGD
SCHEMBL28064841 0.88 ALDH1A1 (0.44) ALDH1A1MEN1GAAMAPTHPGD
SCHEMBL7686914 0.88 HTR7 (0.40) CHRNA7MTNR1BHTR2C
SCHEMBL7684611 0.81 HTR1A (0.43) CHRNA7HTR2C
SCHEMBL7677541 0.81 CHRNA7 (0.42) CHRNA7MTNR1B
SCHEMBL7678362 0.79 SLC6A2 (0.41) CHRNA7MTNR1BHTR2C
SCHEMBL7678292 0.77 CHRNA7 (0.67) CHRNA7HTR2C
SCHEMBL7680425 0.77 CHRNA7 (0.67) CHRNA7HTR2C
SCHEMBL7680070 0.77 CHRNA7 (0.67) CHRNA7HTR2C
SCHEMBL6002146 0.76 HTR1A (0.45) HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6417183-B1 DRUGS RELATES TO 1,4-DIAZACYCLOHEPTANES, TO PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND TO THEIR USE IN METHODS OF THERAPEUTIC TREATMENT OF NERVOUS SYSTEM DISORDERS ASTRAZENELA UK LIMITED (GB) 2002-07-09 US disclosed
EP-1060169-A1 1,4-DIAZACYCLOHEPTANE DERIVATIVES AstraZeneca AB (SE) 2000-12-20 EP disclosed
WO-1999032461-A1 1,4-DIAZACYCLOHEPTANE DERIVATIVES ASTRAZENECA UK LIMITED (GB) 1999-07-01 WO disclosed