SCHEMBL7683116

SCHEMBL7683116

COc1c(S(=O)(=O)Cl)cc(Br)c2ccc(C)nc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.38
KMT2A Q03164 3/20 0.38
HTT P42858 3/20 0.37
PKM P14618 1/20 0.37
GAA P10253 1/20 0.36
ALDH1A1 P00352 3/20 0.36
SLC40A1 Q9NP59 1/20 0.34
TRPV4 Q9HBA0 1/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 2/20 0.33
CCR1 P32246 1/20 0.33
RAB9A P51151 1/20 0.33
CCR5 P51681 1/20 0.33
NSD2 O96028 1/20 0.33
G6PD P11413 1/20 0.33
DNMT1 P26358 1/20 0.33
USP2 O75604 1/20 0.33
POLB P06746 1/20 0.33
TSHR P16473 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7690476 0.79 NQO2 (0.50) KDM4EKMT2AHTTPKMGAA
SCHEMBL7693657 0.78 SMN1; SMN2 (0.45) KDM4EKMT2AHTTALDH1A1LMNA
SCHEMBL7692165 0.73 KDM4E (0.38) KDM4EKMT2AHTTPKMGAA
SCHEMBL13737587 0.68 RAB9A (0.52) KDM4EKMT2AHTTLMNACCR1
SCHEMBL28554817 0.68 KDM4E (0.40) KDM4EKMT2AHTTPKMGAA
SCHEMBL18106122 0.68 KDM4E (0.42) KDM4EKMT2AHTTPKMGAA
SCHEMBL9951347 0.67 KDM4E (0.41) KDM4EKMT2AHTTPKMGAA
SCHEMBL5212965 0.67 NQO2 (0.40) KDM4EKMT2AHTTPKMALDH1A1
SCHEMBL31579147 0.66 TRPV4 (0.43) KDM4EHTTPKMGAAALDH1A1
SCHEMBL7690466 0.66 MAPT (0.67) KDM4EKMT2AHTTPKMGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6500842-B1 N-((4-CHLOROPHENYL)METHYL)-8-HYDROXY-7-QUINOLINECARBOXAMIDE ADMINISTERED AS VIRICIDES AGAINST HERPES VIRUS PHARMACIA & UPJOHN COMPANY 2002-12-31 US disclosed
US-6310211-B1 ANTI-VIRAL ACTIVITY AGAINST HERPES VIRUS, CYTOMEGALOVIRUS. MANY OF THESE COMPOUNDS ARE ALSO ACTIVE AGAINST VARICELLA ZOSTER VIRUS, EPSTEIN-BARR VIRUS, HERPES SIMPLEX VIRUS AND HUMAN HERPES VIRUS TYPE 8 PHARMACIA & UPJOHN COMPANY 2001-10-30 US disclosed
US-6252080-B1 HERPES, CYTOMEGALO VIRUS PHARMACIA & UPJOHN COMPANY 2001-06-26 US disclosed
US-6211376-B1 HERPES VIRUS, CYTOMEGALO VIRUS, VARICELLA-ZOSTER VIRUS,EPSTEIN-BARR VIRUS PHARMACIA & UPJOHN COMPANY 2001-04-03 US disclosed
EP-0927164-A1 8-HYDROXY-7-SUBSTITUTED QUINOLINES AS ANTI-VIRAL AGENTS PHARMACIA & UPJOHN COMPANY (US) 1999-07-07 EP disclosed
WO-1998011073-A1 8-HYDROXY-7-SUBSTITUTED QUINOLINES AS ANTI-VIRAL AGENTS PHARMACIA & UPJOHN COMPANY (US) 1998-03-19 WO disclosed