SCHEMBL7690476

SCHEMBL7690476

COc1c(Br)cc(Br)c2ccc(C)nc12

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 3/20 0.50
RAB9A P51151 2/20 0.42
CCR1 P32246 1/20 0.42
CCR5 P51681 1/20 0.42
CA2 P00918 1/20 0.41
CA4 P22748 1/20 0.41
KDM4E B2RXH2 5/20 0.39
KMT2A Q03164 3/20 0.39
HTT P42858 3/20 0.38
PKM P14618 1/20 0.38
MAPT P10636 4/20 0.37
OPRK1 P41145 1/20 0.36
LMNA P02545 2/20 0.36
MEN1 O00255 1/20 0.36
TLR9 Q9NR96 1/20 0.36
USP2 O75604 1/20 0.36
POLB P06746 1/20 0.36
TSHR P16473 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
ADORA1 P30542 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28554817 0.83 KDM4E (0.40) NQO2RAB9ACCR1CCR5KDM4E
SCHEMBL9951347 0.82 KDM4E (0.41) RAB9ACCR1CCR5KDM4EKMT2A
SCHEMBL13737587 0.80 RAB9A (0.52) NQO2RAB9ACCR1CCR5KDM4E
SCHEMBL18106122 0.80 KDM4E (0.42) RAB9ACCR1CCR5KDM4EKMT2A
SCHEMBL7692165 0.79 KDM4E (0.38) NQO2RAB9ACCR1CCR5KDM4E
SCHEMBL7683116 0.79 KDM4E (0.38) NQO2RAB9ACCR1CCR5KDM4E
SCHEMBL5212965 0.76 NQO2 (0.40) NQO2RAB9ACCR1CCR5KDM4E
Broquinaldol SCHEMBL2110667 0.75 MAPT (0.54) NQO2RAB9ACCR1CCR5KDM4E
Broquinaldol SCHEMBL29606314 0.75 MAPT (0.54) NQO2RAB9ACCR1CCR5KDM4E
Broxaldine SCHEMBL2109050 0.74 ALOX5 (0.41) RAB9ACA2KDM4EKMT2AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6500842-B1 N-((4-CHLOROPHENYL)METHYL)-8-HYDROXY-7-QUINOLINECARBOXAMIDE ADMINISTERED AS VIRICIDES AGAINST HERPES VIRUS PHARMACIA & UPJOHN COMPANY 2002-12-31 US disclosed
US-6310211-B1 ANTI-VIRAL ACTIVITY AGAINST HERPES VIRUS, CYTOMEGALOVIRUS. MANY OF THESE COMPOUNDS ARE ALSO ACTIVE AGAINST VARICELLA ZOSTER VIRUS, EPSTEIN-BARR VIRUS, HERPES SIMPLEX VIRUS AND HUMAN HERPES VIRUS TYPE 8 PHARMACIA & UPJOHN COMPANY 2001-10-30 US disclosed
US-6252080-B1 HERPES, CYTOMEGALO VIRUS PHARMACIA & UPJOHN COMPANY 2001-06-26 US disclosed
US-6211376-B1 HERPES VIRUS, CYTOMEGALO VIRUS, VARICELLA-ZOSTER VIRUS,EPSTEIN-BARR VIRUS PHARMACIA & UPJOHN COMPANY 2001-04-03 US disclosed
EP-0927164-A1 8-HYDROXY-7-SUBSTITUTED QUINOLINES AS ANTI-VIRAL AGENTS PHARMACIA & UPJOHN COMPANY (US) 1999-07-07 EP disclosed
WO-1998011073-A1 8-HYDROXY-7-SUBSTITUTED QUINOLINES AS ANTI-VIRAL AGENTS PHARMACIA & UPJOHN COMPANY (US) 1998-03-19 WO disclosed