SCHEMBL7683193

SCHEMBL7683193

Cc1cc(C)nc(N(C)c2ccccc2I)n1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
C1R P00736 1/20 0.42
ALDH1A1 P00352 5/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
CRHR1 P34998 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
KDM4E B2RXH2 1/20 0.36
HTT P42858 2/20 0.33
LMNA P02545 1/20 0.33
HPGD P15428 1/20 0.33
USP2 O75604 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7687657 0.75 CRHR1 (0.47) ALDH1A1CRHR1
SCHEMBL8034298 0.70 CRHR1 (0.41) ALDH1A1L3MBTL1CRHR1
SCHEMBL12811256 0.69 C1R (0.45) C1RMEN1KMT2AHTT
SCHEMBL3838727 0.67 MAPT (0.44) C1RALDH1A1L3MBTL1KDM4ELMNA
SCHEMBL29893980 0.67 MAPT (0.44) C1RALDH1A1L3MBTL1KDM4ELMNA
SCHEMBL8033081 0.67 CRHR1 (0.46) ALDH1A1CRHR1LMNA
SCHEMBL7680765 0.67 CRHR1 (0.46) L3MBTL1CRHR1
SCHEMBL10879962 0.66 ACHE (0.35) ALDH1A1MAPT
SCHEMBL26756570 0.65 APP (0.38) C1RALDH1A1KDM4EMAPT
SCHEMBL9877961 0.64 TSHR (0.42) ALDH1A1L3MBTL1MEN1KMT2AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6342503-B1 ANTIDEPRESSANTS, EATING DISORDERS DUPONT PHARMACEUTICALS COMPANY 2002-01-29 US disclosed
US-6107301-A PSYCHOLOGICAL DISORDERS DUPONT PHARMACEUTICALS COMPANY (US) 2000-08-22 US disclosed
EP-0723533-A1 1N-ALKYL-N-ARYLPYRIMIDINAMINES AND DERIVATIVES THEREOF THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-07-31 EP disclosed
WO-1995010506-A1 1N-ALKYL-N-ARYLPYRIMIDINAMINES AND DERIVATIVES THEREOF THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-04-20 WO disclosed