SCHEMBL7687657

SCHEMBL7687657

Cc1cc(C)nc(N(C)c2ccccc2C(F)(F)F)n1

nearest known ligand 0.59

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 7/20 0.47
ALDH1A1 P00352 1/20 0.43
TSHR P16473 1/20 0.43
RBP4 P02753 3/20 0.40
ACP1 P24666 1/20 0.40
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CLK4 Q9HAZ1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7683193 0.75 C1R (0.42) CRHR1ALDH1A1
SCHEMBL1935074 0.74 CYP1A2 (0.40) CRHR1ALDH1A1TSHRACP1CYP1A2
SCHEMBL805589 0.73 HSD11B1 (0.51) CRHR1ALDH1A1TSHRCYP1A2CYP2D6
SCHEMBL17479870 0.72 HDAC6 (0.45) ALDH1A1TSHRACP1CYP1A2CYP2D6
SCHEMBL7687275 0.71 CRHR1 (0.43) CRHR1
SCHEMBL1768874 0.70 ACP1 (0.46) ALDH1A1TSHRACP1CYP1A2CYP2D6
SCHEMBL30454780 0.70 ACP1 (0.46) ALDH1A1TSHRACP1CYP1A2CYP2D6
SCHEMBL9737393 0.70 ALDH1A1 (0.43) CRHR1ALDH1A1TSHRRBP4
SCHEMBL1935076 0.68 CYP1A2 (0.40) ALDH1A1TSHRACP1CYP1A2CYP2D6
SCHEMBL2093130 0.67 ESR1 (0.38) ALDH1A1TSHRACP1CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6342503-B1 ANTIDEPRESSANTS, EATING DISORDERS DUPONT PHARMACEUTICALS COMPANY 2002-01-29 US disclosed
US-6107301-A PSYCHOLOGICAL DISORDERS DUPONT PHARMACEUTICALS COMPANY (US) 2000-08-22 US disclosed
WO-1995010506-A1 1N-ALKYL-N-ARYLPYRIMIDINAMINES AND DERIVATIVES THEREOF THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-04-20 WO disclosed