SCHEMBL7683232

SCHEMBL7683232

Oc1ccc(C2(c3ccc(Br)cc3)CC2)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 8/20 0.64
ESR1 P03372 7/20 0.64
ALOX15 P16050 2/20 0.59
GLB1 P16278 1/20 0.46
CTRB1 P17538 1/20 0.46
CTRC Q99895 1/20 0.46
AGER Q15109 1/20 0.38
ALDH1A1 P00352 3/20 0.36
KDM4E B2RXH2 2/20 0.36
MAPT P10636 2/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
NPC1 O15118 1/20 0.36
CA12 O43570 1/20 0.36
GMNN O75496 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
LMNA P02545 1/20 0.36
CA3 P07451 1/20 0.36
CYP3A4 P08684 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14260454 0.90 ESR1 (0.80) ESR2ESR1ALOX15GLB1CTRB1
SCHEMBL7530533 0.88 ESR2 (0.80) ESR2ESR1ALOX15ALDH1A1KDM4E
SCHEMBL3811364 0.88 ESR2 (0.80) ESR2ESR1ALOX15ALDH1A1KDM4E
SCHEMBL1977810 0.86 ESR1 (0.53) ESR2ESR1ALOX15GLB1CTRB1
SCHEMBL31540169 0.86 ESR2 (0.53) ESR2ESR1ALOX15GLB1CTRB1
SCHEMBL9838333 0.81 ESR2 (0.95) ESR2ESR1ALOX15ALDH1A1KDM4E
SCHEMBL19428169 0.81 ESR2 (0.70) ESR2ESR1ALOX15ALDH1A1KDM4E
SCHEMBL23198889 0.79 OPRM1 (0.52) ESR2ESR1ALDH1A1MEN1KMT2A
SCHEMBL14804313 0.79 OPRM1 (0.52) ESR2ESR1ALDH1A1MEN1KMT2A
SCHEMBL14804316 0.79 OPRM1 (0.52) ESR2ESR1ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6441177-B1 Tertiary amines HOFFMANN-LA ROCHE INC. 2002-08-27 US disclosed
EP-0778264-B1 Tertiary amines having antimycotic and cholesterol lowering activity HOFFMANN LA ROCHE (CH) 2001-07-11 EP disclosed
US-6034275-A FUGICIDES; ATICHOLESTEROL AGENTS HOFFMANN-LA ROCHE INC. (US) 2000-03-07 US disclosed
CN-1158844-A Tertiary amines HOFFMANN LA ROCHE (CH) 1997-09-10 CN disclosed
EP-0778264-A1 Tertiary amines having antimycotic and cholesterol lowering activity F. HOFFMANN-LA ROCHE AG (CH) 1997-06-11 EP disclosed