SCHEMBL7683483

SCHEMBL7683483

Cc1cnc(Nc2nc(C)cc(C)n2)c(Br)c1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.47
ALDH1A1 P00352 2/20 0.47
POLB P06746 2/20 0.40
KDM4E B2RXH2 2/20 0.40
CYP1A2 P05177 3/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
LMNA P02545 1/20 0.39
NPC1 O15118 4/20 0.38
RAB9A P51151 4/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
TP53 P04637 1/20 0.38
AHR P35869 1/20 0.36
ADORA2A P29274 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15426468 0.74 MAPT (0.37) MAPTALDH1A1KDM4ECYP1A2CYP3A4
SCHEMBL3942497 0.72 IGF1R (0.50) ALDH1A1KDM4ECYP1A2CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL28381933 0.72 MAPT (0.36) MAPTALDH1A1KDM4ECYP1A2CYP2D6
SCHEMBL3940988 0.71 ALDH1A1 (0.50) MAPTALDH1A1CYP1A2MEN1KMT2A
SCHEMBL3940864 0.71 MAPT (0.41) MAPTALDH1A1CYP1A2NPC1RAB9A
SCHEMBL7684971 0.70 MAPT (0.67) MAPTALDH1A1LMNANPC1RAB9A
SCHEMBL3947432 0.70 KDM4E (0.34) MAPTALDH1A1KDM4E
SCHEMBL3941768 0.70 MAPK10 (0.44) KDM4ELMNANPC1RAB9AMEN1
SCHEMBL17492679 0.70 AURKA (0.44) MAPTALDH1A1POLBCYP1A2CYP3A4
SCHEMBL22853792 0.70 LMNA (0.64) MAPTALDH1A1KDM4ECYP1A2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6342503-B1 ANTIDEPRESSANTS, EATING DISORDERS DUPONT PHARMACEUTICALS COMPANY 2002-01-29 US disclosed
US-6107301-A PSYCHOLOGICAL DISORDERS DUPONT PHARMACEUTICALS COMPANY (US) 2000-08-22 US disclosed
EP-0723533-A1 1N-ALKYL-N-ARYLPYRIMIDINAMINES AND DERIVATIVES THEREOF THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-07-31 EP disclosed
WO-1995010506-A1 1N-ALKYL-N-ARYLPYRIMIDINAMINES AND DERIVATIVES THEREOF THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-04-20 WO disclosed