Itaconate

Itaconate

SCHEMBL7683801

C=C(CC(=O)O)C(=O)O.CCC(C)(C)OC=Cc1ccccc1

nearest known ligand 0.39

Full drug profile on Sugi Atlas →

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
EGFR P00533 4/20 0.38
ALOX15 P16050 1/20 0.37
HSD17B10 Q99714 1/20 0.37
HAO1 Q9UJM8 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HDAC3 O15379 1/20 0.36
CTDSP1 Q9GZU7 1/20 0.36
PAM P19021 1/20 0.36
RECQL P46063 1/20 0.35
CYP2C19 P33261 1/20 0.35
NPC1 O15118 3/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
RAB9A P51151 3/20 0.34
LMNA P02545 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
PPARA Q07869 1/20 0.34
KMT2A Q03164 1/20 0.34
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3783785 0.82 RELA (0.43) EGFRALOX15HSD17B10ALDH1A1CYP2C19
SCHEMBL27414917 0.72 HAO1 (0.44) EGFRHAO1ALDH1A1HDAC3PAM
Itaconate SCHEMBL11309982 0.72 MEN1 (0.48) EGFRHAO1ALDH1A1HDAC3CTDSP1
Itaconate SCHEMBL3201278 0.71 ALOX15 (0.57) ALOX15HSD17B10HAO1ALDH1A1HDAC3
Juarezic Acid SCHEMBL8768055 0.70 HDAC3 (0.53) ALOX15HSD17B10HAO1ALDH1A1HDAC3
Itaconate SCHEMBL6053436 0.70 ALOX15 (0.47) ALOX15HSD17B10HAO1ALDH1A1HDAC3
SCHEMBL9128813 0.70 CYP2C19 (0.41) EGFRALDH1A1HDAC3CTDSP1PAM
Itaconate SCHEMBL7058781 0.69 ALOX15 (0.44) ALOX15HSD17B10ALDH1A1RECQLCYP2C19
SCHEMBL8401214 0.69 PPARA (0.43) EGFRHAO1ALDH1A1HDAC3CTDSP1
Itaconate SCHEMBL11140941 0.68 ALOX15 (0.42) ALOX15HSD17B10HAO1ALDH1A1HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6395367-B1 ELECTROCONDUCTIVITY HYDRO-QUEBEC (CA) 2002-05-28 US claimed