SCHEMBL7684485

SCHEMBL7684485

CC1=CC(C)(C)N(c2cccc(F)c2F)c2ccccc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.47
ALDH1A1 P00352 7/20 0.46
NPSR1 Q6W5P4 5/20 0.46
GAA P10253 2/20 0.46
TSHR P16473 2/20 0.43
USP2 O75604 1/20 0.43
MAPK1 P28482 1/20 0.43
MAPT P10636 6/20 0.41
KMT2A Q03164 5/20 0.41
KDM4E B2RXH2 4/20 0.41
MCOLN3 Q8TDD5 1/20 0.39
MEN1 O00255 4/20 0.36
HPGD P15428 1/20 0.35
HTT P42858 1/20 0.35
PGR P06401 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CRHBP P24387 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27512034 0.76 NPSR1 (0.47) LMNAALDH1A1NPSR1GAATSHR
SCHEMBL27512035 0.76 LMNA (0.47) LMNAALDH1A1NPSR1GAATSHR
SCHEMBL9724434 0.73 NPSR1 (0.55) LMNAALDH1A1NPSR1GAATSHR
SCHEMBL28226781 0.72 LMNA (0.56) LMNAALDH1A1NPSR1GAATSHR
SCHEMBL28312197 0.72 LMNA (0.46) LMNAALDH1A1NPSR1GAATSHR
SCHEMBL8871090 0.71 NPSR1 (0.48) LMNAALDH1A1NPSR1GAATSHR
SCHEMBL27476136 0.71 NPSR1 (0.44) LMNAALDH1A1NPSR1GAATSHR
SCHEMBL2393621 0.70 LMNA (0.57) LMNAALDH1A1NPSR1GAATSHR
SCHEMBL29367208 0.69 LMNA (0.53) LMNAALDH1A1NPSR1GAATSHR
SCHEMBL8832558 0.69 NPSR1 (0.43) LMNAALDH1A1NPSR1GAATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1175247-A Steroid receptor modulator compounds and methods LIGAND PHARM INC (US) 1998-03-04 CN claimed
US-6448405-B1 COUPLING A 2-HALO-5-NITROBENZOIC ACID AND A 2-METHOXYPHENYL BORONIC ACID; CYCLIZING TO A NITROBENZOCOUMARIN; REDUCING TO THE AMINE; CONVERTING TO A COUMARINO(3,4-F)QUINOLINE; REDUCTION TO A 5H-CHROMENO(3,4-F)QUINOLINE LIGAND PHARMACEUTICALS INCORPORATED 2002-09-10 US disclosed