Cyclopropane

Cyclopropane

SCHEMBL7686540

C1CC1.CN(c1ccc(F)cc1)c1ccc(F)cc1

nearest known ligand 0.46

Full drug profile on Sugi Atlas →

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
APP P05067 2/20 0.46
SLC6A4 P31645 2/20 0.42
SLC6A3 Q01959 2/20 0.42
SLC6A2 P23975 1/20 0.42
CES1 P23141 1/20 0.42
ACHE P22303 1/20 0.39
TAAR1 Q96RJ0 1/20 0.38
DDB1 Q16531 1/20 0.38
CRBN Q96SW2 1/20 0.38
TRPA1 O75762 1/20 0.38
TSHR P16473 2/20 0.36
ALDH1A1 P00352 2/20 0.36
ALOX15 P16050 1/20 0.36
HSD17B10 Q99714 1/20 0.36
AOC3 Q16853 1/20 0.35
MPO P05164 1/20 0.35
SIGMAR1 Q99720 1/20 0.34
KCNH2 Q12809 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13338132 0.92 APP (0.52) APPCES1ACHETAAR1DDB1
Cyclopropane SCHEMBL28538522 0.84 APP (0.64) APPSLC6A4SLC6A3SLC6A2TSHR
SCHEMBL20800879 0.82 SLC18A3 (0.41) APPDDB1CRBNTRPA1ALDH1A1
SCHEMBL20800882 0.82 ACHE (0.65) APPCES1ACHETAAR1TSHR
SCHEMBL307380 0.82 CES1 (0.49) APPSLC6A4SLC6A2CES1TSHR
SCHEMBL25354186 0.80 APP (0.43) APPCES1ACHETAAR1DDB1
SCHEMBL20800878 0.80 SLC18A3 (0.42) APPDDB1CRBNTRPA1ALDH1A1
SCHEMBL5998627 0.78 CHRM5 (0.52) APPSLC6A2CES1TAAR1ALOX15
SCHEMBL10031935 0.78 APP (0.76) APPALOX15KCNH2
SCHEMBL22681645 0.78 RXRA (0.41) APPSLC6A4SLC6A3SLC6A2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001096283-A9 HIV INTEGRASE INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2002-10-17 WO disclosed