SCHEMBL7687463

SCHEMBL7687463

N#Cc1ccc(C(=O)c2ccc(OC/C=C/CBr)c(F)c2)cc1

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 2/20 0.40
VNN1 O95497 5/20 0.38
P4HB P07237 2/20 0.38
GAA P10253 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
ACHE P22303 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
AR P10275 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7687468 1.00 GSK3B (0.40) GSK3BVNN1P4HBGAASMN1; SMN2
SCHEMBL8047384 0.85 LSS (0.43) ACHEALDH1A1MAPT
SCHEMBL8904544 0.85 LSS (0.43) ACHEALDH1A1MAPT
SCHEMBL8905081 0.82 ALDH1A1 (0.49) GSK3BVNN1ALDH1A1MAPT
SCHEMBL8047800 0.82 ALDH1A1 (0.49) GSK3BVNN1ALDH1A1MAPT
SCHEMBL7685849 0.81 F10 (0.39) VNN1AR
SCHEMBL8903738 0.81 ACHE (0.36) ACHE
SCHEMBL8044773 0.81 ACHE (0.36) ACHE
SCHEMBL7685855 0.80 LSS (0.57) VNN1GAASMN1; SMN2ACHE
SCHEMBL7685852 0.80 LSS (0.57) VNN1GAASMN1; SMN2ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6441177-B1 Tertiary amines HOFFMANN-LA ROCHE INC. 2002-08-27 US disclosed
EP-0778264-B1 Tertiary amines having antimycotic and cholesterol lowering activity HOFFMANN LA ROCHE (CH) 2001-07-11 EP disclosed
EP-0636367-B1 Use of phenylalkylamines for producing cholesterol lowering agents HOFFMANN LA ROCHE (CH) 2000-03-29 EP disclosed
US-6034275-A FUGICIDES; ATICHOLESTEROL AGENTS HOFFMANN-LA ROCHE INC. (US) 2000-03-07 US disclosed
EP-0778264-A1 Tertiary amines having antimycotic and cholesterol lowering activity F. HOFFMANN-LA ROCHE AG (CH) 1997-06-11 EP disclosed
US-5637771-A Compound useful for lowering cholesterol HOFFMANN-LA ROCHE INC. (US) 1997-06-10 US disclosed
US-5574071-A ADMINISTERING PHENYLALKYLAMINO KETONES HOFFMANN-LA ROCHE INC. (US) 1996-11-12 US disclosed
US-5495048-A ANTICHOLESTEROL AGENTS HOFFMANN-LA ROCHE INC. (US) 1996-02-27 US disclosed
EP-0636367-A1 Use of phenylalkylamines for producing cholesterol lowering agents F. HOFFMANN-LA ROCHE AG (CH) 1995-02-01 EP disclosed