SCHEMBL8047800

SCHEMBL8047800

N#Cc1ccc(C(=O)c2ccc(OC/C=C/CBr)cc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.49
MAPT P10636 1/20 0.49
GSK3B P49841 2/20 0.47
LSS P48449 3/20 0.46
VNN1 O95497 2/20 0.44
PARP15 Q460N3 1/20 0.44
PARP10 Q53GL7 1/20 0.44
PARP2 Q9UGN5 1/20 0.44
RAB9A P51151 1/20 0.44
MMP2 P08253 2/20 0.41
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
MMP1 P03956 1/20 0.39
MMP3 P08254 1/20 0.39
MMP9 P14780 1/20 0.39
MMP13 P45452 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8905081 1.00 ALDH1A1 (0.49) ALDH1A1MAPTGSK3BLSSVNN1
SCHEMBL1714552 0.88 MAOB (0.44) ALDH1A1MAPTGSK3BMMP2CA1
SCHEMBL1714549 0.88 MAOB (0.44) ALDH1A1MAPTGSK3BMMP2CA1
SCHEMBL9360157 0.84 GAA (0.55) ALDH1A1MAPTLSSRAB9A
SCHEMBL7685512 0.84 LSS (0.62) MAPTLSSRAB9A
SCHEMBL9360152 0.84 GAA (0.55) ALDH1A1MAPTLSSRAB9A
SCHEMBL7685521 0.84 LSS (0.62) MAPTLSSRAB9A
SCHEMBL7687468 0.82 GSK3B (0.40) ALDH1A1MAPTGSK3BVNN1
SCHEMBL7687463 0.82 GSK3B (0.40) ALDH1A1MAPTGSK3BVNN1
SCHEMBL8902853 0.82 LSS (0.48) ALDH1A1MAPTLSSPARP10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0636367-B1 Use of phenylalkylamines for producing cholesterol lowering agents HOFFMANN LA ROCHE (CH) 2000-03-29 EP disclosed
US-5637771-A Compound useful for lowering cholesterol HOFFMANN-LA ROCHE INC. (US) 1997-06-10 US disclosed
US-5574071-A ADMINISTERING PHENYLALKYLAMINO KETONES HOFFMANN-LA ROCHE INC. (US) 1996-11-12 US disclosed
US-5495048-A ANTICHOLESTEROL AGENTS HOFFMANN-LA ROCHE INC. (US) 1996-02-27 US disclosed
EP-0636367-A1 Use of phenylalkylamines for producing cholesterol lowering agents F. HOFFMANN-LA ROCHE AG (CH) 1995-02-01 EP disclosed