SCHEMBL7688546

SCHEMBL7688546

CS(=O)(=O)NCC(=O)[C@H](Cc1ccccc1)NC(=O)c1ccccc1NS(=O)(=O)c1ccc2ccccc2c1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 6/20 0.46
BCL2 P10415 1/20 0.46
BCL2L1 Q07817 1/20 0.46
MCL1 Q07820 1/20 0.46
BCL2A1 Q16548 1/20 0.46
SLC16A3 O15427 2/20 0.44
CCKAR P32238 2/20 0.43
CCKBR P32239 2/20 0.43
PLAT P00750 1/20 0.43
F2 P00734 1/20 0.43
KAT6A Q92794 1/20 0.43
KEAP1 Q14145 1/20 0.42
NFE2L2 Q16236 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7695356 0.87 SLC16A3 (0.48) KCNA5BCL2BCL2L1MCL1BCL2A1
SCHEMBL7706585 0.85 ALDH1A1 (0.53) PLATF2KAT6A
SCHEMBL7694179 0.84 AKR1C3 (0.48) SLC16A3PLATF2KAT6A
SCHEMBL7422050 0.80 KCNA5 (0.49) KCNA5KAT6A
SCHEMBL7786988 0.80 BCL2 (0.51) KCNA5BCL2BCL2L1MCL1BCL2A1
SCHEMBL7786990 0.80 BCL2 (0.51) KCNA5BCL2BCL2L1MCL1BCL2A1
SCHEMBL7694857 0.80 CA2 (0.43) KCNA5CCKARCCKBRKAT6A
SCHEMBL7791340 0.79 CAPN1 (0.60) KCNA5BCL2BCL2L1MCL1BCL2A1
SCHEMBL7384115 0.79 CAPN1 (0.60) KCNA5BCL2BCL2L1MCL1BCL2A1
SCHEMBL7703492 0.79 CA2 (0.42) CCKARCCKBRPLAT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6436925-B1 BETTER ABLE TO CROSS MEMBRANES; INHIBITORS OF CYSTEINE PROTEASES LIKE CALPAIN I AND II AND CATHEPSIN B AND L, CAN THUS BE USED TO CONTROL DISEASES ASSOCIATED WITH AN ELEVATED ACTIVITY OF CALPAIN ENZYMES OR CATHEPSIN ENZYMES ABBOTT LABORATORIES 2002-08-20 US disclosed