SCHEMBL7703492

SCHEMBL7703492

Cc1cc(Nc2ccc3ccccc3c2)ccc1C(=O)N[C@@H](Cc1ccccc1)C(=O)CNS(C)(=O)=O

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CA2 P00918 3/20 0.42
L3MBTL1 Q9Y468 1/20 0.40
CAPN1 P07384 1/20 0.39
CTSL P07711 1/20 0.39
CTSB P07858 1/20 0.39
KMT2A Q03164 1/20 0.39
ITGB1 P05556 2/20 0.39
ITGA4 P13612 2/20 0.39
PIN1 Q13526 1/20 0.39
PLAT P00750 1/20 0.39
CCKAR P32238 1/20 0.39
CCKBR P32239 1/20 0.39
ACE P12821 2/20 0.38
CA1 P00915 1/20 0.38
MMP2 P08253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7702126 0.91 PLAT (0.45) CA2L3MBTL1PLATCCKARCCKBR
SCHEMBL7698087 0.90 CA2 (0.51) CA2CTSLCTSBKMT2APIN1
SCHEMBL7706585 0.81 ALDH1A1 (0.53) CA2KMT2APLATCA1
SCHEMBL7694857 0.80 CA2 (0.43) CA2CAPN1CTSLCTSBPIN1
SCHEMBL7429916 0.79 MAPK9 (0.41) CA2CCKBRACE
SCHEMBL7700700 0.79 CA2 (0.52) CA2CTSLCTSBKMT2AITGB1
SCHEMBL7688546 0.79 KCNA5 (0.46) PLATCCKARCCKBR
SCHEMBL7421589 0.79 PYGL (0.43) CA2PLATCCKBRACE
SCHEMBL7420454 0.78 PYGL (0.33)
SCHEMBL7690013 0.77 CAPN1 (0.68) CA2CAPN1CTSLCTSBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6436925-B1 BETTER ABLE TO CROSS MEMBRANES; INHIBITORS OF CYSTEINE PROTEASES LIKE CALPAIN I AND II AND CATHEPSIN B AND L, CAN THUS BE USED TO CONTROL DISEASES ASSOCIATED WITH AN ELEVATED ACTIVITY OF CALPAIN ENZYMES OR CATHEPSIN ENZYMES ABBOTT LABORATORIES 2002-08-20 US disclosed