SCHEMBL7689499

SCHEMBL7689499

Cc1cn(C)c2c1C(=O)CC(c1ccccc1)C2

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.47
HSP90AA1 P07900 1/20 0.46
HSP90AB1 P08238 1/20 0.46
TSHR P16473 3/20 0.45
ALOX15 P16050 1/20 0.45
HSD17B10 Q99714 1/20 0.45
KMT2A Q03164 5/20 0.44
MEN1 O00255 4/20 0.44
ALDH1A1 P00352 3/20 0.44
CSNK2A2 P19784 2/20 0.44
CSNK2B P67870 2/20 0.44
CSNK2A1 P68400 2/20 0.44
ABCG2 Q9UNQ0 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
HPGD P15428 3/20 0.44
MAP1LC3B Q9GZQ8 1/20 0.43
CASP1 P29466 1/20 0.43
CASP7 P55210 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL27523012 0.81 MEN1 (0.36) LMNAHSP90AA1HSP90AB1TSHRKMT2A
SCHEMBL7686746 0.81 LMNA (0.43) LMNAHSP90AA1HSP90AB1TSHRALOX15
SCHEMBL16797470 0.77 KDM4E (0.42) LMNAHSP90AA1HSP90AB1TSHRALOX15
SCHEMBL7686928 0.74 MAP1LC3B (0.50) LMNATSHRKMT2AMEN1ALDH1A1
Hydrochloric Acid SCHEMBL7685341 0.71 HPGD (0.34) LMNAHSD17B10HPGD
SCHEMBL7685368 0.69 LMNA (0.58) LMNAHSP90AA1HSP90AB1TSHRALOX15
SCHEMBL7685234 0.69 ALOX15 (0.56) LMNAHSP90AA1HSP90AB1TSHRALOX15
SCHEMBL7687667 0.68 CSNK2A2 (0.44) LMNAHSP90AA1HSP90AB1TSHRALOX15
SCHEMBL7685559 0.67 HSP90AA1 (0.61) LMNAHSP90AA1HSP90AB1TSHRALOX15
SCHEMBL14959525 0.67 BRD4 (0.67) TSHRKMT2AMEN1ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6350749-B1 SODIUM CHANNEL MODULATORS, ANTIARRHYTHMIA AND HYPOTENSIVE AGENTS; CARDIOVASCULAR DISORDERS, ANGINA PECTORIS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-02-26 US disclosed
EP-1057812-A1 AMINOGUANIDINE HYDRAZONE DERIVATIVES, PROCESS FOR PRODUCING THE SAME AND DRUGS THEREOF Takeda Chemical Industries, Ltd. (JP) 2000-12-06 EP disclosed