SCHEMBL7689583

SCHEMBL7689583

COC(=O)c1ccc(NC(=O)c2ccc(Cl)[nH]c2=O)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 8/20 0.54
MEN1 O00255 7/20 0.54
RAB9A P51151 5/20 0.50
SMN1; SMN2 Q16637 5/20 0.50
NPC1 O15118 4/20 0.50
HTT P42858 3/20 0.50
ATM Q13315 1/20 0.50
TAS1R3 Q7RTX0 1/20 0.50
TAS1R1 Q7RTX1 1/20 0.50
GAA P10253 1/20 0.50
PTPN1 P18031 1/20 0.48
ALDH1A1 P00352 4/20 0.47
HPGD P15428 2/20 0.47
KDM4E B2RXH2 2/20 0.47
LMNA P02545 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
CRHBP P24387 1/20 0.47
CYP2C19 P33261 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31032981 0.79 KDM4E (0.66) RAB9ASMN1; SMN2NPC1HTTATM
SCHEMBL21639567 0.74 EGFR (0.54) KMT2AMEN1RAB9ASMN1; SMN2NPC1
SCHEMBL6263820 0.74 NPC1 (0.83) KMT2AMEN1RAB9ASMN1; SMN2NPC1
SCHEMBL8660366 0.74 NPC1 (0.83) KMT2AMEN1RAB9ASMN1; SMN2NPC1
SCHEMBL7690950 0.74 PPARG (0.56) KMT2AMEN1RAB9ANPC1HTT
SCHEMBL21242859 0.73 NPC1 (0.71) KMT2AMEN1RAB9ASMN1; SMN2NPC1
SCHEMBL15444796 0.72 HTT (0.55) KMT2AMEN1RAB9ASMN1; SMN2NPC1
SCHEMBL10272284 0.71 MEN1 (0.74) KMT2AMEN1ALDH1A1HPGDKDM4E
SCHEMBL15917720 0.71 MEN1 (0.61) KMT2AMEN1RAB9ASMN1; SMN2NPC1
SCHEMBL25349531 0.71 MEN1 (0.65) KMT2AMEN1SMN1; SMN2PTPN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002053544-A1 PHARMACEUTICAL USES AND SYNTHESIS OF NICOTINANILIDE-N-OXIDES DARWIN DISCOVERY LTD. (GB) 2002-07-11 WO disclosed