SCHEMBL7689802

SCHEMBL7689802

Cc1ccc(Cl)c(C2CC(=O)CC(=O)C2)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.59
RECQL P46063 1/20 0.59
MAPT P10636 2/20 0.39
GAA P10253 1/20 0.39
MAPK1 P28482 1/20 0.36
BRD4 O60885 1/20 0.36
CREBBP Q92793 1/20 0.36
CHRNB2 P17787 1/20 0.35
CHRNA4 P43681 1/20 0.35
POLB P06746 1/20 0.35
KMT2A Q03164 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
THRB P10828 1/20 0.35
ACHE P22303 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
ALDH1A1 P00352 1/20 0.34
ALDH2 P05091 1/20 0.34
PBRM1 Q86U86 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7560192 0.82 TP53 (0.44) TP53RECQLMAPTGAACHRNB2
SCHEMBL7685669 0.82 TP53 (0.62) TP53RECQLMAPTGAACHRNB2
SCHEMBL30558904 0.79 TP53 (0.42) TP53RECQLMAPTGAABRD4
SCHEMBL6796450 0.79 TP53 (0.59) TP53RECQLMAPTGAACHRNB2
SCHEMBL7685976 0.79 TP53 (0.42) TP53RECQLMAPTGAACHRNB2
SCHEMBL23625888 0.79 TP53 (0.49) TP53RECQLMAPK1CHRNB2CHRNA4
SCHEMBL13454023 0.79 GRM7 (0.47) TP53RECQLMAPTGAACHRNB2
SCHEMBL13454044 0.78 TP53 (0.41) TP53RECQLMAPTGAACHRNB2
SCHEMBL13806045 0.77 CHRNB2 (0.41) CHRNB2CHRNA4
SCHEMBL7690082 0.76 POLB (0.36) TP53RECQLMAPK1BRD4CREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6350749-B1 SODIUM CHANNEL MODULATORS, ANTIARRHYTHMIA AND HYPOTENSIVE AGENTS; CARDIOVASCULAR DISORDERS, ANGINA PECTORIS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-02-26 US disclosed
EP-1057812-A1 AMINOGUANIDINE HYDRAZONE DERIVATIVES, PROCESS FOR PRODUCING THE SAME AND DRUGS THEREOF Takeda Chemical Industries, Ltd. (JP) 2000-12-06 EP disclosed
EP-0950418-A2 Composition for preventing or treating ischemic disease Takeda Chemical Industries, Ltd. (JP) 1999-10-20 EP disclosed