SCHEMBL7685976

SCHEMBL7685976

Cc1ccc(F)c(C2CC(=O)CC(=O)C2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.42
RECQL P46063 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.40
TDP1 Q9NUW8 2/20 0.40
MAPT P10636 2/20 0.39
GAA P10253 1/20 0.39
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
MAOB P27338 1/20 0.35
KMT2A Q03164 3/20 0.35
NPSR1 Q6W5P4 3/20 0.35
CHRNB2 P17787 1/20 0.35
CHRNA4 P43681 1/20 0.35
POLB P06746 1/20 0.35
ACHE P22303 1/20 0.34
HTR1A P08908 1/20 0.34
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
SLC6A3 Q01959 1/20 0.34
MEN1 O00255 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6794027 0.82 KDM1A (0.46) TP53RECQLTDP1MAPTGAA
SCHEMBL7560192 0.82 TP53 (0.44) TP53RECQLTDP1MAPTGAA
SCHEMBL7683113 0.81 TP53 (0.51) TP53RECQLL3MBTL1TDP1MAPT
SCHEMBL7689802 0.79 TP53 (0.59) TP53RECQLTDP1MAPTGAA
SCHEMBL30558904 0.79 TP53 (0.42) TP53RECQLTDP1MAPTGAA
SCHEMBL13454023 0.79 GRM7 (0.47) TP53RECQLTDP1MAPTGAA
SCHEMBL13454044 0.78 TP53 (0.41) TP53RECQLTDP1MAPTGAA
SCHEMBL12024476 0.77 SLC6A2 (0.45) L3MBTL1TDP1CA1CA2CHRNB2
SCHEMBL7689625 0.76 L3MBTL1 (0.47) L3MBTL1TDP1KMT2ANPSR1POLB
SCHEMBL10452140 0.74 ALDH1A1 (0.47) TP53RECQLMAPTKMT2ACHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6350749-B1 SODIUM CHANNEL MODULATORS, ANTIARRHYTHMIA AND HYPOTENSIVE AGENTS; CARDIOVASCULAR DISORDERS, ANGINA PECTORIS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-02-26 US disclosed
EP-1057812-A1 AMINOGUANIDINE HYDRAZONE DERIVATIVES, PROCESS FOR PRODUCING THE SAME AND DRUGS THEREOF Takeda Chemical Industries, Ltd. (JP) 2000-12-06 EP disclosed