SCHEMBL769210

SCHEMBL769210

COCNC(=O)C1CCOc2ccccc21

nearest known ligand 0.57

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SSTR4 P31391 1/20 0.44
P2RX7 Q99572 8/20 0.43
HPGD P15428 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
MAPT P10636 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25463803 0.85 SSTR4 (0.46) SSTR4P2RX7HPGDMAPTKMT2A
SCHEMBL23985230 0.83 HTR2B (0.48) SSTR4P2RX7HPGDMAPTKMT2A
SCHEMBL5846881 0.80 SSTR4 (0.43) SSTR4SMN1; SMN2KMT2A
SCHEMBL29724343 0.80 SSTR4 (0.43) SSTR4SMN1; SMN2KMT2A
SCHEMBL25112123 0.80 SSTR4 (0.46) SSTR4P2RX7SMN1; SMN2
SCHEMBL5846877 0.80 SSTR4 (0.43) SSTR4SMN1; SMN2KMT2A
SCHEMBL5846872 0.80 SSTR4 (0.43) SSTR4SMN1; SMN2KMT2A
SCHEMBL24897847 0.77 ITGAV (0.45) SSTR4P2RX7HPGDSMN1; SMN2L3MBTL1
SCHEMBL24897846 0.75 SSTR4 (0.45) SSTR4P2RX7HPGDL3MBTL1MAPT
SCHEMBL769529 0.75 PRMT5 (0.52) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120071506-A1 METHODS FOR TREATING CNS DISORDERS WITH BICYCLO-SUBSTITUTED 2-IMIDAZOLINE AND 2-IMIDAZOLES GALLEY GUIDO (DE) 2012-03-22 US disclosed
EP-1981499-A1 USE OF 2-IMIDAZOLES FOR THE TREATMENT OF CNS DISORDERS F.HOFFMANN-LA ROCHE AG (CH) 2008-10-22 EP disclosed
US-20070197620-A1 Methods for treating CNS disorders with bicyclo-substituted 2-imidazoline and 2-imidazoles HOFFMANN-LA ROCHE INC. 2007-08-23 US disclosed
WO-2007085558-A1 USE OF 2-IMIDAZOLES FOR THE TREATMENT OF CNS DISORDERS F. HOFFMANN-LA ROCHE AG (CH) 2007-08-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120071506-A1 METHODS FOR TREATING CNS DISORDERS WITH BICYCLO-SUBSTITUTED 2-IMIDAZOLINE AND 2-IMIDAZOLES CRY1, PER2, GPR119 SSTR4 593/4885P2RX7 248/4885HPGD 4058/4885
US-20070197620-A1 Methods for treating CNS disorders with bicyclo-substituted 2-imidazoline and 2-imidazoles CRY1, PER2, GPR119 SSTR4 555/4885P2RX7 250/4885HPGD 3748/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.