SCHEMBL7696004

SCHEMBL7696004

O=C(N[C@@H](Cc1ccccc1)C(=O)CNS(=O)(=O)c1ccccc1)c1ccccc1C=Cc1ccccn1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 12/20 0.46
CTSB P07858 8/20 0.46
CTSL P07711 4/20 0.43
CASP1 P29466 1/20 0.43
CTSS P25774 4/20 0.41
CTSK P43235 2/20 0.41
USP30 Q70CQ3 1/20 0.41
KCNA5 P22460 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7698037 0.90 CAPN1 (0.47) CAPN1CTSBCTSLCTSSCTSK
SCHEMBL7689922 0.88 CAPN1 (0.57) CAPN1CTSBCTSLCASP1CTSS
SCHEMBL7693964 0.87 CAPN1 (0.50) CAPN1CTSBCTSLCASP1CTSS
SCHEMBL7695268 0.86 CTSB (0.44) CAPN1CTSBCASP1CTSSCTSK
SCHEMBL7693583 0.84 CAPN1 (0.48) CAPN1CTSBCTSLCTSSCTSK
SCHEMBL7696533 0.84 CAPN1 (0.48) CAPN1CTSBCTSLCTSSCTSK
SCHEMBL7705654 0.83 CAPN1 (0.46) CAPN1CTSBCTSLCASP1CTSS
SCHEMBL7698802 0.82 CAPN1 (0.67) CAPN1CTSBCTSLCASP1CTSS
SCHEMBL7688501 0.80 CAPN1 (0.58) CAPN1CTSBCTSLCASP1CTSS
SCHEMBL7695839 0.79 CAPN1 (0.70) CAPN1CTSBCTSLCASP1CTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6436925-B1 BETTER ABLE TO CROSS MEMBRANES; INHIBITORS OF CYSTEINE PROTEASES LIKE CALPAIN I AND II AND CATHEPSIN B AND L, CAN THUS BE USED TO CONTROL DISEASES ASSOCIATED WITH AN ELEVATED ACTIVITY OF CALPAIN ENZYMES OR CATHEPSIN ENZYMES ABBOTT LABORATORIES 2002-08-20 US disclosed