SCHEMBL7698079

SCHEMBL7698079

COc1cc(C2CO2)ccc1O[Si](c1ccccc1)(c1ccccc1)C(C)(C)C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.40
MAPK3 P27361 1/20 0.40
MAPK1 P28482 1/20 0.40
HTR2C P28335 1/20 0.38
PTAFR P25105 1/20 0.38
ALOX5 P09917 1/20 0.37
PTPN1 P18031 1/20 0.37
PPARG P37231 1/20 0.37
PPARD Q03181 1/20 0.37
ALDH1A1 P00352 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
TSHR P16473 1/20 0.36
GAA P10253 2/20 0.36
RAB9A P51151 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
PDE4A P27815 1/20 0.35
PDE4B Q07343 1/20 0.35
PDE4C Q08493 1/20 0.35
PDE4D Q08499 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6257872 0.76 NPC1 (0.36) MAPK1HTR2CALDH1A1MEN1KMT2A
SCHEMBL30108108 0.76 NR3C2 (0.40) HTR2CMEN1KMT2A
SCHEMBL4709625 0.76 MAPT (0.46) MAPK1HTR2CALDH1A1MEN1KMT2A
SCHEMBL5334814 0.76 NPC1 (0.43) MAPK1ALDH1A1MEN1KMT2ATSHR
SCHEMBL26507116 0.76 NR3C2 (0.40) HTR2CMEN1KMT2A
SCHEMBL6257880 0.76 NQO2 (0.34) MAPK1HTR2CALDH1A1MEN1KMT2A
SCHEMBL901629 0.76 ACHE (0.57) ACHEMAPK3MAPK1PTAFRALOX5
SCHEMBL7700239 0.75 HTR2C (0.35) HTR2CALDH1A1MEN1KMT2AGAA
SCHEMBL5331625 0.73 ENPP2 (0.36) RAB9A
SCHEMBL31737879 0.73 ENPP2 (0.36) RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002006229-A2 HETEROCYCLIC BETA-3 ADRENERGIC RECEPTOR AGONISTS WYETH (US) 2002-01-24 WO disclosed